Small molecule positive allosteric modulation of TRPV1 activation by vanilloids and acidic pH.
about
Positive allosteric modulation of TRPV1 as a novel analgesic mechanism.Molecular Surgery Concept from Bench to Bedside: A Focus on TRPV1+ Pain-Sensing Neurons.Targeting breast cancer cells by MRS1477, a positive allosteric modulator of TRPV1 channels.Affimer proteins are versatile and renewable affinity reagentsNociception and inflammatory hyperalgesia evaluated in rodents using infrared laser stimulation after Trpv1 gene knockout or resiniferatoxin lesionConstrained TRPV1 agonists synthesized via silver-mediated intramolecular azo-methine ylide cycloaddition of α-iminoamides.A systematic review of the association between immunogenomic markers and cancer-related fatigueBlockade of transient receptor potential cation channel subfamily V member 1 promotes regeneration after sciatic nerve injury.Vanilloids selectively sensitize thermal glutamate release from TRPV1 expressing solitary tract afferentsResiniferatoxin for Pain Treatment: An Interventional Approach to Personalized Pain Medicine.The fundamental unit of pain is the cell.Altered pharmacology of native rodent spinal cord TRPV1 after phosphorylation.TRPV1 antagonist capsazepine suppresses 4-AP-induced epileptiform activity in vitro and electrographic seizures in vivo.Effect of TRPV1 channel on the proliferation and apoptosis in asthmatic rat airway smooth muscle cells.Investigating the involvement of TRPV1 ion channels in remote hind limb preconditioning-induced cardioprotection in rats.TRPV1 antagonists that cause hypothermia, instead of hyperthermia, in rodents: compounds' pharmacological profiles, in-vivo targets, thermoeffectors recruited, and implications for drug development.Pain control through selective chemo-axotomy of centrally projecting TRPV1+ sensory neurons.
P2860
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P2860
Small molecule positive allosteric modulation of TRPV1 activation by vanilloids and acidic pH.
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
2011年论文
@zh
2011年论文
@zh-cn
name
Small molecule positive allost ...... n by vanilloids and acidic pH.
@ast
Small molecule positive allost ...... n by vanilloids and acidic pH.
@en
type
label
Small molecule positive allost ...... n by vanilloids and acidic pH.
@ast
Small molecule positive allost ...... n by vanilloids and acidic pH.
@en
prefLabel
Small molecule positive allost ...... n by vanilloids and acidic pH.
@ast
Small molecule positive allost ...... n by vanilloids and acidic pH.
@en
P2093
P2860
P356
P1476
Small molecule positive allost ...... on by vanilloids and acidic pH
@en
P2093
Claudio Coddou
Jason M Keller
Krisztian Kaszas
Mark A Hoon
Michael J Iadarola
Santosh K Mishra
Stanko Stojilkovic
P2860
P304
P356
10.1124/JPET.111.183053
P407
P577
2011-10-17T00:00:00Z