Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
about
CNS active O-linked glycopeptidesOpioid peptidomimetics: leads for the design of bioavailable mixed efficacy μ opioid receptor (MOR) agonist/δ opioid receptor (DOR) antagonist ligandsCan amphipathic helices influence the CNS antinociceptive activity of glycopeptides related to β-endorphin?Development of a bioavailable μ opioid receptor (MOPr) agonist, δ opioid receptor (DOPr) antagonist peptide that evokes antinociception without development of acute tolerance.The development of biomarkers to reduce attrition rate in drug discovery focused on oncology and central nervous system.Translation of structure-activity relationships from cyclic mixed efficacy opioid peptides to linear analoguesIn Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt(1)-DALDA Analogues.Comparing naturally occurring glycosylated forms of proline rich antibacterial peptide, Drosocin.
P2860
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P2860
Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
description
2012 nî lūn-bûn
@nan
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
2012年论文
@zh
2012年论文
@zh-cn
name
Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
@ast
Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
@en
type
label
Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
@ast
Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
@en
prefLabel
Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
@ast
Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
@en
P2093
P2860
P356
P1476
Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins
@en
P2093
Dhanasekaran Muthu
Edward J Bilsky
Jean M Bidlack
Mark R Lefever
Robin Polt
Yingxue Li
P2860
P304
P356
10.4155/FMC.11.195
P577
2012-02-01T00:00:00Z