Search for new purine- and ribose-modified adenosine analogues as selective agonists and antagonists at adenosine receptors
about
Purine (N)-Methanocarba Nucleoside Derivatives Lacking an Exocyclic Amine as Selective A3 Adenosine Receptor Agonists.A3-adenosine receptors: design of selective ligands and therapeutic prospectsStructure-based approaches to ligands for G-protein-coupled adenosine and P2Y receptors, from small molecules to nanoconjugates.N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors.Adenosine receptor agonists: from basic medicinal chemistry to clinical development.Rigidified A3 Adenosine Receptor Agonists: 1-Deazaadenine Modification Maintains High in Vivo EfficacyEFA (9-beta-D-erythrofuranosyladenine) is an effective salvage agent for methylthioadenosine phosphorylase-selective therapy of T-cell acute lymphoblastic leukemia with L-alanosine.Induction of apoptosis in HL-60 human promyelocytic leukemia cells by adenosine A(3) receptor agonists.Medicinal chemistry of the A3 adenosine receptor: agonists, antagonists, and receptor engineering.Structure-activity relationships of 9-alkyladenine and ribose-modified adenosine derivatives at rat A3 adenosine receptors.Methanocarba analogues of purine nucleosides as potent and selective adenosine receptor agonists.Novel approaches for targeting the adenosine A2A receptor.Determination and validation of LJ-2698, a potent human A3 adenosine receptor antagonist, in rat plasma by liquid chromatography-tandem mass spectrometry and its application in pharmacokinetic study.Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonist.Deoxy Derivatives of L-like 5'-Noraristeromycin.A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy.Adenosine A3 receptor and brain. A culprit, a hero, or merely yet another receptor?Synthesis of carbocyclic 2-substituted adenine nucleoside and related analogs.
P2860
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P2860
Search for new purine- and ribose-modified adenosine analogues as selective agonists and antagonists at adenosine receptors
description
1995 nî lūn-bûn
@nan
1995年の論文
@ja
1995年学术文章
@wuu
1995年学术文章
@zh-cn
1995年学术文章
@zh-hans
1995年学术文章
@zh-my
1995年学术文章
@zh-sg
1995年學術文章
@yue
1995年學術文章
@zh
1995年學術文章
@zh-hant
name
Search for new purine- and rib ...... gonists at adenosine receptors
@ast
Search for new purine- and rib ...... gonists at adenosine receptors
@en
type
label
Search for new purine- and rib ...... gonists at adenosine receptors
@ast
Search for new purine- and rib ...... gonists at adenosine receptors
@en
prefLabel
Search for new purine- and rib ...... gonists at adenosine receptors
@ast
Search for new purine- and rib ...... gonists at adenosine receptors
@en
P2093
P2860
P356
P1476
Search for new purine- and rib ...... gonists at adenosine receptors
@en
P2093
G Cristalli
J A Secrist
K A Jacobson
K N Tiwari
S M Siddiqi
S W Schneller
P2860
P304
P356
10.1021/JM00007A014
P407
P577
1995-03-01T00:00:00Z