Design, synthesis, and SAR studies of 4-substituted methoxylbenzoyl-aryl-thiazoles analogues as potent and orally bioavailable anticancer agents
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Novel Natural Product- and Privileged Scaffold-Based Tubulin Inhibitors Targeting the Colchicine Binding SiteCurrent Advances of Tubulin Inhibitors in Nanoparticle Drug Delivery and Vascular Disruption/AngiogenesisIdentification of diaryl 5-amino-1,2,4-oxadiazoles as tubulin inhibitors: the special case of 3-(2-fluorophenyl)-5-(4-methoxyphenyl)amino-1,2,4-oxadiazoleSystemic delivery of nanoparticle formulation of novel tubulin inhibitor for treating metastatic melanoma.Palladium-catalyzed arylation of cyanamides.Palladium-catalyzed N-arylation of 2-aminothiazolesStructural Optimization of Indole Derivatives Acting at Colchicine Binding Site as Potential Anticancer Agents2-Substituted 4,5-dihydrothiazole-4-carboxylic acids are novel inhibitors of metallo-β-lactamasesOrally bioavailable tubulin antagonists for paclitaxel-refractory cancer.New substituted 4H-chromenes as anticancer agents.Discovery and Optimization of N-Substituted 2-(4-pyridinyl)thiazole carboxamides against Tumor Growth through Regulating Angiogenesis Signaling Pathways.Diaryl and heteroaryl sulfides: synthesis via sulfenyl chlorides and evaluation as selective anti-breast-cancer agents.Synthesis and cellular uptake of p-[(123)I]-phenyl-amino-thiazole ((123)I-PAT) as a potential agent for targeting tubulin polymerization in tumors.Formulation and characterization of polyester/polycarbonate nanoparticles for delivery of a novel microtubule destabilizing agentDiscovery of novel 2-aryl-4-benzoyl-imidazole (ABI-III) analogues targeting tubulin polymerization as antiproliferative agents.Efficient synthesis of novel 3-aryl-5-(4-chloro-2-morpholinothiazol-5-yl)-4,5-dihydro-1H-pyrazoles and their antifungal activity alone and in combination with commercial antifungal agents.Cell penetrating thiazole peptides inhibit c-MYC expression via site-specific targeting of c-MYC G-quadruplex.
P2860
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P2860
Design, synthesis, and SAR studies of 4-substituted methoxylbenzoyl-aryl-thiazoles analogues as potent and orally bioavailable anticancer agents
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
2011年论文
@zh
2011年论文
@zh-cn
name
Design, synthesis, and SAR stu ...... bioavailable anticancer agents
@ast
Design, synthesis, and SAR stu ...... bioavailable anticancer agents
@en
type
label
Design, synthesis, and SAR stu ...... bioavailable anticancer agents
@ast
Design, synthesis, and SAR stu ...... bioavailable anticancer agents
@en
prefLabel
Design, synthesis, and SAR stu ...... bioavailable anticancer agents
@ast
Design, synthesis, and SAR stu ...... bioavailable anticancer agents
@en
P2093
P2860
P356
P1476
Design, synthesis, and SAR stu ...... bioavailable anticancer agents
@en
P2093
Chien-Ming Li
Duane D Miller
Jianjun Chen
Michael L Mohler
P2860
P304
P356
10.1021/JM2003427
P407
P577
2011-06-07T00:00:00Z