ATP-dependent uptake of natural product cytotoxic drugs by membrane vesicles establishes MRP as a broad specificity transporter.
about
Anthrapyridones, a novel group of antitumour non-cross resistant anthraquinone analogues. Synthesis and molecular basis of the cytotoxic activity towards K562/DOX cells.Modeling the chemoprotective functions of glutathione S-transferases in cultured cell lines by heterologous expression.Metabolic engineering of plant cells in a space environment.Hepatic glutathione and glutathione S-conjugate transport mechanismsThe role of drug efflux pumps in acute myeloid leukemia.Inhibition of the MRP1-mediated transport of the menadione-glutathione conjugate (thiodione) in HeLa cells as studied by SECM.Modulation of oral drug bioavailability: from preclinical mechanism to therapeutic application.The prognostic significance of expression of the multidrug resistance-associated protein (MRP) in primary breast cancerCytotoxicity of rhein, the active metabolite of sennoside laxatives, is reduced by multidrug resistance-associated protein 1The ability of selected pyridinium salts to increase the cytotoxic activity of vincristine but not doxorubicin towards sensitive and multidrug resistant promyelocytic leukaemia HL60 cells.Indomethacin induces apoptosis via a MRP1-dependent mechanism in doxorubicin-resistant small-cell lung cancer cells overexpressing MRP1.Development and characterization of multidrug resistant human hepatocarcinoma cell line in nude mice.The role of bioreductive activation of doxorubicin in cytotoxic activity against leukaemia HL60-sensitive cell line and its multidrug-resistant sublines.The human multidrug-resistance-associated protein MRP1 mediates ATP-dependent transport of unconjugated bilirubinATP-dependent transport of reduced glutathione in yeast secretory vesicles.Resolution of P-glycoprotein and non-P-glycoprotein effects on drug permeability using intestinal tissues from mdr1a (-/-) mice.ATPase activity of purified multidrug resistance-associated protein.Functional expression of P-glycoprotein and multidrug resistance-associated protein (Mrp1) in primary cultures of rat astrocytes.ATP-dependent transport of reduced glutathione on YCF1, the yeast orthologue of mammalian multidrug resistance associated proteins.
P2860
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P2860
ATP-dependent uptake of natural product cytotoxic drugs by membrane vesicles establishes MRP as a broad specificity transporter.
description
article científic
@ca
article scientifique
@fr
articolo scientifico
@it
artigo científico
@pt
bilimsel makale
@tr
scientific article published on July 1996
@en
vedecký článok
@sk
vetenskaplig artikel
@sv
videnskabelig artikel
@da
vědecký článek
@cs
name
ATP-dependent uptake of natura ...... broad specificity transporter.
@en
ATP-dependent uptake of natura ...... broad specificity transporter.
@nl
type
label
ATP-dependent uptake of natura ...... broad specificity transporter.
@en
ATP-dependent uptake of natura ...... broad specificity transporter.
@nl
prefLabel
ATP-dependent uptake of natura ...... broad specificity transporter.
@en
ATP-dependent uptake of natura ...... broad specificity transporter.
@nl
P2093
P2860
P356
P1476
ATP-dependent uptake of natura ...... broad specificity transporter.
@en
P2093
P2860
P304
P356
10.1073/PNAS.93.14.6929
P407
P577
1996-07-01T00:00:00Z