PET radioligands for the vesicular acetylcholine transporter (VAChT).
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SLC transporters as therapeutic targets: emerging opportunitiesThe Concise Guide to PHARMACOLOGY 2013/14: transporters.Synthesis and labeling of a piperazine-based library of ¹¹C-labeled ligands for imaging of the vesicular acetylcholine transporter.A new VGLUT-specific potent inhibitor: pharmacophore of Brilliant YellowIdentification and characterization of ML352: a novel, noncompetitive inhibitor of the presynaptic choline transporter.In vitro and ex vivo characterization of (-)-TZ659 as a ligand for imaging the vesicular acetylcholine transporterSynthesis and biological characterization of a promising F-18 PET tracer for vesicular acetylcholine transporter.Synthesis and evaluation of in vitro bioactivity for vesicular acetylcholine transporter inhibitors containing two carbonyl groups.Automated production of [¹⁸F]VAT suitable for clinical PET study of vesicular acetylcholine transporter.Kinetics modeling and occupancy studies of a novel C-11 PET tracer for VAChT in nonhuman primates.Heteroaromatic and aniline derivatives of piperidines as potent ligands for vesicular acetylcholine transporter.Development of (18)F-labeled radiotracers for neuroreceptor imaging with positron emission tomographyIn vitro and in vivo characterization of two C-11-labeled pet tracers for vesicular acetylcholine transporter.Syntheses and radiosyntheses of two carbon-11 labeled potent and selective radioligands for imaging vesicular acetylcholine transporter.A Numbering System for MFS Transporter Proteins.Concordance between in vivo and postmortem measurements of cholinergic denervation in rats using PET with [18F]FEOBV and choline acetyltransferase immunochemistry.Bio-orthogonal labeling as a tool to visualize and identify newly synthesized proteins in Caenorhabditis elegans.Synthesis, resolution, and in vitro evaluation of three vesicular acetylcholine transporter ligands and evaluation of the lead fluorine-18 radioligand in a nonhuman primate.Development of novel PET probe [¹¹C](R,R)HAPT and its stereoisomer [¹¹C](S,S)HAPT for vesicular acetylcholine transporter imaging: a PET study in conscious monkey.In Vivo and In Vitro Characteristics of Radiolabeled Vesamicol Analogs as the Vesicular Acetylcholine Transporter Imaging Agents.
P2860
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P2860
PET radioligands for the vesicular acetylcholine transporter (VAChT).
description
article científic
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article scientifique
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articolo scientifico
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artigo científico
@pt
bilimsel makale
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scientific article published on January 2010
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vedecký článok
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vetenskaplig artikel
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videnskabelig artikel
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vědecký článek
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name
PET radioligands for the vesicular acetylcholine transporter (VAChT).
@en
PET radioligands for the vesicular acetylcholine transporter
@nl
type
label
PET radioligands for the vesicular acetylcholine transporter (VAChT).
@en
PET radioligands for the vesicular acetylcholine transporter
@nl
prefLabel
PET radioligands for the vesicular acetylcholine transporter (VAChT).
@en
PET radioligands for the vesicular acetylcholine transporter
@nl
P2093
P1476
PET radioligands for the vesicular acetylcholine transporter (VAChT).
@en
P2093
Aurélie Boucher-Arnold
Ian Mat Som
Michael Kassiou
Nicolas Giboureau
P304
P356
10.2174/156802610793176846
P577
2010-01-01T00:00:00Z