En route to new blockbuster anti-histamines: surveying the offspring of the expanding histamine receptor family.
about
Histamine and Skin Barrier: Are Histamine Antagonists Useful for the Prevention or Treatment of Atopic Dermatitis?Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readoutsHistamine H3 receptor antagonists/inverse agonists on cognitive and motor processes: relevance to Alzheimer's disease, ADHD, schizophrenia, and drug abuseThe Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsDesign and pharmacological characterization of VUF14480, a covalent partial agonist that interacts with cysteine 98(3.36) of the human histamine H₄ receptor.LC-MS/MS method for the determination of pitolisant: application to rat pharmacokinetic and brain penetration studies.Regulation of mammalian physiology, development, and disease by the sphingosine 1-phosphate and lysophosphatidic acid receptors.Regulation of mast cell responses in health and disease.Effects of methimepip and JNJ-5207852 in Wistar rats exposed to an open-field with and without object and in Balb/c mice exposed to a radial-arm mazeCombinatorial roles for histamine H1-H2 and H3-H4 receptors in autoimmune inflammatory disease of the central nervous system.Preclinical evaluation of the abuse potential of Pitolisant, a histamine H₃ receptor inverse agonist/antagonist compared with ModafinilMolecular and cellular analysis of human histamine receptor subtypes.Several down, a few to go: histamine H3 receptor ligands making the final push towards the market?Biogenic amines and the control of neuromuscular signaling in schistosomes.Histamine H3 receptor antagonists in relation to epilepsy and neurodegeneration: a systemic consideration of recent progress and perspectives.Procognitive properties of drugs with single and multitargeting H3 receptor antagonist activities.Development of a profiling strategy for metabolic mixtures by combining chromatography and mass spectrometry with cell-based GPCR signaling.A structural chemogenomics analysis of aminergic GPCRs: lessons for histamine receptor ligand design.Commercially available antibodies against human and murine histamine H₄-receptor lack specificity.Interactions of recombinant human histamine H₁R, H₂R, H₃R, and H₄R receptors with 34 antidepressants and antipsychotics.Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology.Structure-based virtual screening for fragment-like ligands of the G protein-coupled histamine H4 receptor
P2860
Q26799561-C7C47E96-E507-4647-8768-2AFC6882DCC8Q28536518-B8862FE2-97DD-430C-8760-126FDD0163B7Q30462161-6F4D041D-01A7-414F-9938-B7EF81D46F9EQ30486707-E5D1E4FE-11AD-4CED-A0BF-362D3B63425BQ34324177-0438C496-A27D-48B1-A721-2989C4295496Q34769004-62F51127-E972-4717-98CC-934D5B461B0BQ35551835-399F73F1-2667-4959-8D3A-8B09737EFD89Q36092456-6340F9C8-74B2-4C7C-B4BD-13C99336FA1DQ36096591-38BDB8E6-9AD1-46A8-A291-A34BCE673DB2Q36430032-048C99F1-6CA5-4270-AC0F-29F0DC15B630Q36929453-17597EEE-7358-4DE4-808E-A439FE70753DQ37407709-190DC4FC-0654-4B99-883F-F62C16DED128Q37944920-E753BB80-F1EA-417D-9931-025B85305AACQ38004814-16AC73E8-B716-4427-9FA9-D6B3C490E5C6Q38023551-BD2CEF05-D555-4DD6-93B5-8A72A1772919Q38212433-B7F30E54-D200-4B0A-86A4-573C1BD76E25Q39323929-2B470AC9-F4A7-4249-8D8B-1F63F9BFD747Q39411714-C463E353-04EC-47FA-B3AA-4E5212B2C3D2Q39445688-563F55C6-1581-423B-BEA4-3BDCD78064C8Q48812098-2A1E5D9B-AC12-42A1-A20B-6FD122892600Q55232052-3257C9EE-252F-49B2-9FBC-FBD227FE8E36Q56991394-16F41FB3-4FBF-4B6B-A8B5-A4250C7778DD
P2860
En route to new blockbuster anti-histamines: surveying the offspring of the expanding histamine receptor family.
description
article científic
@ca
article scientifique
@fr
articolo scientifico
@it
artigo científico
@pt
bilimsel makale
@tr
scientific article published on 15 March 2011
@en
vedecký článok
@sk
vetenskaplig artikel
@sv
videnskabelig artikel
@da
vědecký článek
@cs
name
En route to new blockbuster an ...... ing histamine receptor family.
@en
En route to new blockbuster an ...... ing histamine receptor family.
@nl
type
label
En route to new blockbuster an ...... ing histamine receptor family.
@en
En route to new blockbuster an ...... ing histamine receptor family.
@nl
prefLabel
En route to new blockbuster an ...... ing histamine receptor family.
@en
En route to new blockbuster an ...... ing histamine receptor family.
@nl
P2093
P1476
En route to new blockbuster an ...... ing histamine receptor family.
@en
P2093
Henry F Vischer
Iwan J P de Esch
Maikel Wijtmans
P304
P356
10.1016/J.TIPS.2011.02.004
P577
2011-03-15T00:00:00Z