Inhibition of aminopeptidases by amastatin and bestatin derivatives. Effect of inhibitor structure on slow-binding processes.
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Leucine aminopeptidase: bestatin inhibition and a model for enzyme-catalyzed peptide hydrolysisCD13 (human aminopeptidase N) mediates human cytomegalovirus infectionA Role for the Brain RAS in Alzheimer's and Parkinson's DiseasesBinding structure of the leucine aminopeptidase inhibitor microginin FR1Synthesis of New (−)-Bestatin-Based Inhibitor Libraries Reveals a Novel Binding Mode in the S1 Pocket of the Essential Malaria M1 MetalloaminopeptidaseBestatin-based chemical biology strategy reveals distinct roles for malaria M1- and M17-family aminopeptidasesThe X-ray Crystal Structure of Human Aminopeptidase N Reveals a Novel Dimer and the Basis for Peptide ProcessingNovel and highly sensitive fluorescent assay for leucine aminopeptidasesCharacterization of peptide fluxes into human erythrocytes. A proton-n.m.r. studyDevelopment of novel assays for proteolytic enzymes using rhodamine-based fluorogenic substrates.Development of Synthetic Aminopeptidase N/CD13 Inhibitors to Overcome Cancer Metastasis and Angiogenesis.In vivo imaging of leucine aminopeptidase activity in drug-induced liver injury and liver cancer via a near-infrared fluorescent probe.Effects of tachykinins on uterine smooth muscle.Proteins of the kidney microvillar membrane. Enzymic and molecular properties of aminopeptidase WStructural basis for the inhibition of M1 family aminopeptidases by the natural product actinonin: Crystal structure in complex with E. coli aminopeptidase N.Angiotensin induction of PAI-1 expression in endothelial cells is mediated by the hexapeptide angiotensin IVNeuropeptide degrading enzymes in normal and inflamed human synovium.Characterization of the tachykinin NK2 receptor in the human bronchus: influence of amastatin-sensitive metabolic pathwaysIntestinal peptidases form functional complexes with the neutral amino acid transporter B(0)AT1.Identification of alanyl aminopeptidase (CD13) as a surface marker for isolation of mature gastric zymogenic chief cells.Inhibition of tryptase release from human colon mast cells by protease inhibitors.Modulation of histamine release from human colon mast cells by protease inhibitors.Angiotensin receptor subtype mediated physiologies and behaviors: new discoveries and clinical targets.Aminopeptidase N (EC 3.4.11.2) inhibitors (2006 - 2010): a patent review.The brain renin-angiotensin system: a diversity of functions and implications for CNS diseases.A glutamate residue contributes to the exopeptidase specificity in aminopeptidase AThe Extracellular Vesicles of the Helminth Pathogen, Fasciola hepatica: Biogenesis Pathways and Cargo Molecules Involved in Parasite Pathogenesis.Angiotensin-III is Increased in Alzheimer's Disease in Association with Amyloid-β and Tau Pathology.Design, synthesis and biological evaluation of novel L-isoserine tripeptide derivatives as aminopeptidase N inhibitors.Design, synthesis and preliminary activity evaluation of novel 3-amino-2-hydroxyl-3-phenylpropanoic acid derivatives as aminopeptidase N/CD13 inhibitors.Focus on Brain Angiotensin III and Aminopeptidase A in the Control of Hypertension.Inhibition of aminopeptidase M by alkyl D-cysteinates.Cysteinyl-glycine in the control of glutathione homeostasis in bovine lenses.Biochemical characterization of aminopeptidase N2 from Toxoplasma gondii.Development of bestatin-based activity-based probes for metallo-aminopeptidases.Metabolism of neuropeptides. Hydrolysis of the angiotensins, bradykinin, substance P and oxytocin by pig kidney microvillar membranes.Ethanol modulates neuropeptide-degrading aminopeptidases at synapse level in calcium-dependent conditions.Ectoenzymes of the kidney microvillar membrane. Affinity purification, characterization and localization of the phospholipase C-solubilized form of renal dipeptidase.Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.Design and synthesis of substrate-based inhibitors of botulinum neurotoxin type B metalloprotease.
P2860
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P2860
Inhibition of aminopeptidases by amastatin and bestatin derivatives. Effect of inhibitor structure on slow-binding processes.
description
1984 nî lūn-bûn
@nan
1984年の論文
@ja
1984年論文
@yue
1984年論文
@zh-hant
1984年論文
@zh-hk
1984年論文
@zh-mo
1984年論文
@zh-tw
1984年论文
@wuu
1984年论文
@zh
1984年论文
@zh-cn
name
Inhibition of aminopeptidases ...... ure on slow-binding processes.
@en
type
label
Inhibition of aminopeptidases ...... ure on slow-binding processes.
@en
prefLabel
Inhibition of aminopeptidases ...... ure on slow-binding processes.
@en
P2093
P356
P1476
Inhibition of aminopeptidases ...... ure on slow-binding processes.
@en
P2093
P304
P356
10.1021/JM00370A001
P407
P577
1984-04-01T00:00:00Z