Structure-activity relationships of boronic acid inhibitors of dipeptidyl peptidase IV. 1. Variation of the P2 position of Xaa-boroPro dipeptides.
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Epoxomicin, a potent and selective proteasome inhibitor, exhibits in vivo antiinflammatory activityThe Dipeptidyl Peptidase Family, Prolyl Oligopeptidase, and Prolyl Carboxypeptidase in the Immune System and Inflammatory Disease, Including AtherosclerosisIdentification of selective and potent inhibitors of fibroblast activation protein and prolyl oligopeptidasePhase I trial of PT-100 (PT-100), a cytokine-inducing small molecule, following chemotherapy for solid tumor malignancy.Selective inhibition of fibroblast activation protein protease based on dipeptide substrate specificity.Using substrate specificity of antiplasmin-cleaving enzyme for fibroblast activation protein inhibitor design.Phase II assessment of talabostat and cisplatin in second-line stage IV melanoma.Sphingosine kinase 1 isoform-specific interactions in breast cancerDevelopment of Practical Methodologies for the Synthesis of Functionalized Benzoboroxoles.A method for the deprotection of alkylpinacolyl boronate esters.Dipeptidyl-peptidase IV from bench to bedside: an update on structural properties, functions, and clinical aspects of the enzyme DPP IV.Cleavage Specificity of Mycobacterium tuberculosis ClpP1P2 Protease and Identification of Novel Peptide Substrates and Boronate Inhibitors with Anti-bacterial Activity.Talabostat.Peptide and Peptide-Like Modulators of 20S Proteasome Enzymatic Activity in Cancer CellsInhibitor of DASH proteases affects expression of adhesion molecules in osteoclasts and reduces myeloma growth and bone disease.Therapeutic potential of boron-containing compounds.Aminoboronic acids and esters: from synthetic challenges to the discovery of unique classes of enzyme inhibitors.Synthesis of α-aminoboronic acids.DPP8 and DPP9 inhibition induces pro-caspase-1-dependent monocyte and macrophage pyroptosis.Selective fluorescence probes for dipeptidyl peptidase activity-fibroblast activation protein and dipeptidyl peptidase IV.Alzheimer's disease: correlation of the suppression of beta-amyloid peptide secretion from cultured cells with inhibition of the chymotrypsin-like activity of the proteasome.Characterization of peptidyl boronic acid inhibitors of mammalian 20 S and 26 S proteasomes and their inhibition of proteasomes in cultured cellsFibroblast activation protein-α in fibrogenic disorders and cancer: more than a prolyl-specific peptidase?The versatility of boron in biological target engagement.Pyroptosis and Apoptosis Pathways Engage in Bidirectional Crosstalk in Monocytes and Macrophages.
P2860
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P2860
Structure-activity relationships of boronic acid inhibitors of dipeptidyl peptidase IV. 1. Variation of the P2 position of Xaa-boroPro dipeptides.
description
1996 nî lūn-bûn
@nan
1996年の論文
@ja
1996年論文
@yue
1996年論文
@zh-hant
1996年論文
@zh-hk
1996年論文
@zh-mo
1996年論文
@zh-tw
1996年论文
@wuu
1996年论文
@zh
1996年论文
@zh-cn
name
Structure-activity relationshi ...... ion of Xaa-boroPro dipeptides.
@en
Structure-activity relationshi ...... ion of Xaa-boroPro dipeptides.
@nl
type
label
Structure-activity relationshi ...... ion of Xaa-boroPro dipeptides.
@en
Structure-activity relationshi ...... ion of Xaa-boroPro dipeptides.
@nl
prefLabel
Structure-activity relationshi ...... ion of Xaa-boroPro dipeptides.
@en
Structure-activity relationshi ...... ion of Xaa-boroPro dipeptides.
@nl
P2093
P356
P1476
Structure-activity relationshi ...... ion of Xaa-boroPro dipeptides.
@en
P2093
Bachovchin WW
Campbell SJ
Freeman DM
Kennedy CA
Krolikowski DA
Ksiazek JF
P304
P356
10.1021/JM950732F
P407
P577
1996-05-01T00:00:00Z