Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.

Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.

Item
http://www.wikidata.org/entity/Q39366925
Synthesis and evaluation of translocator 18 kDa protein (TSPO) positron emission tomography (PET) radioligands with low binding sensitivity to human single nucleotide polymorphism rs6971.Identification of N-{[6-chloro-4-(2,6-dimethoxyphenyl)quinazolin-2-yl]carbonyl}-l-leucine (NTRC-808), a novel nonpeptide chemotype selective for the neurotensin receptor type 2Long lasting MDM2/Translocator protein modulator: a new strategy for irreversible apoptosis of human glioblastoma cells.Apoptosis therapy in cancer: the first single-molecule co-activating p53 and the translocator protein in glioblastoma.Residence Time, a New parameter to Predict Neurosteroidogenic Efficacy of Translocator Protein (TSPO) Ligands: the Case Study of N,N-Dialkyl-2-arylindol-3-ylglyoxylamides.11C-ER176, a Radioligand for 18-kDa Translocator Protein, Has Adequate Sensitivity to Robustly Image All Three Affinity Genotypes in Human Brain.Translocator protein (TSPO) ligands for the diagnosis or treatment of neurodegenerative diseases: a patent review (2010-2015; part 1).Bridging Pharmaceutical Chemistry with Drug and Nanoparticle Targeting to Investigate the Role of the 18-kDa Translocator Protein TSPO.Transformation of masked benzyl alcohols to o-aminobenzaldehydes through C-H activation: a facile approach to quinazolines.Some insights into the binding mechanism of the GABAA receptor: a combined docking and MM-GBSA study.
P2860

Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.

Item
http://www.wikidata.org/entity/Q39366925
description
2012 nî lūn-bûn
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2012年の論文
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2012年学术文章
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2012年学术文章
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2012年学术文章
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2012年学术文章
@zh-my
2012年学术文章
@zh-sg
2012年學術文章
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2012年學術文章
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2012年學術文章
@zh-hant
name
Synthesis and biological evalu ...... s of the translocator protein.
@en
Synthesis and biological evalu ...... s of the translocator protein.
@nl
type
label
Synthesis and biological evalu ...... s of the translocator protein.
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Synthesis and biological evalu ...... s of the translocator protein.
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prefLabel
Synthesis and biological evalu ...... s of the translocator protein.
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Synthesis and biological evalu ...... s of the translocator protein.
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P1433
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P2093
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P433
P478
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P5875
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P921
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P1476
Synthesis and biological evalu ...... s of the translocator protein.
@en
P2093
P304
P31
P356
P407
P433
P478
P50
P577
P5875
P698
P921