Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
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Synthesis of the thapsigarginsComparison of current docking tools for the simulation of inhibitor binding by the transmembrane domain of the sarco/endoplasmic reticulum calcium ATPasePhosphorylation at threonine-654 is not required for negative regulation of the epidermal growth factor receptor by non-phorbol tumor promoters.Regulation of Ca2+ signaling with particular focus on mast cells.Engineering a prostate-specific membrane antigen-activated tumor endothelial cell prodrug for cancer therapy.The physiological function of store-operated calcium entryAnalysis of the stimulative effect of thapsigargin, a non-TPA-type tumour promoter, on arachidonic acid metabolism in rat peritoneal macrophagesEffects of high-affinity inhibitors on partial reactions, charge movements, and conformational States of the Ca2+ transport ATPase (sarco-endoplasmic reticulum Ca2+ ATPase)Mipsagargin, a novel thapsigargin-based PSMA-activated prodrug: results of a first-in-man phase I clinical trial in patients with refractory, advanced or metastatic solid tumours.Small molecule inhibition of PAX3-FOXO1 through AKT activation suppresses malignant phenotypes of alveolar rhabdomyosarcomaScalable Synthesis of (-)-Thapsigargin.Thapsigargin, a tumor promoter, discharges intracellular Ca2+ stores by specific inhibition of the endoplasmic reticulum Ca2(+)-ATPase.Targeting thapsigargin towards tumors.Arsenic inhibits mast cell degranulation via suppression of early tyrosine phosphorylation events.The functions of store-operated calcium channels.The ability of thapsigargin and thapsigargicin to activate cells involved in the inflammatory response.A novel tumour promoter, thapsigargin, transiently increases cytoplasmic free Ca2+ without generation of inositol phosphates in NG115-401L neuronal cells.Design, synthesis, and biological evaluation of hydroquinone derivatives as novel inhibitors of the sarco/endoplasmic reticulum calcium ATPase.Enhancement by cyclo-oxygenase inhibitors of platelet-activating factor production in thapsigargin-stimulated macrophages.Agonist-induced inhibition of phosphatidylserine synthesis is secondary to the emptying of intracellular Ca2+ stores in Jurkat T-cells.Drug Interactions With the Ca2+-ATPase From Sarco(Endo)Plasmic Reticulum (SERCA).Use of a temporary immersion bioreactor system for the sustainable production of thapsigargin in shoot cultures of
P2860
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P2860
Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
description
1978 nî lūn-bûn
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1978年の論文
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1978年学术文章
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1978年学术文章
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1978年学术文章
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1978年学术文章
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1978年学术文章
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1978年學術文章
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1978年學術文章
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Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
@en
Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
@nl
type
label
Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
@en
Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
@nl
prefLabel
Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
@en
Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
@nl
P2093
P1476
Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L.
@en
P2093
Brøogger Christensen S
Rasmussen U
Sandberg F
P304
P577
1978-01-01T00:00:00Z