Synthesis and biological testing of novel pyridoisothiazolones as histone acetyltransferase inhibitors.
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Structure of a Ternary Naa50p (NAT5/SAN) N-terminal Acetyltransferase Complex Reveals the Molecular Basis for Substrate-specific AcetylationEpigenetic changes modulate schistosome egg formation and are a novel target for reducing transmission of schistosomiasisHistone acetyltransferase inhibitors block neuroblastoma cell growth in vivoSmall molecule inhibitors of histone acetyltransferases as epigenetic tools and drug candidates.Epigenetic control of gene function in schistosomes: a source of therapeutic targets?Analysis of structure-based virtual screening studies and characterization of identified active compounds.High throughput screening identifies modulators of histone deacetylase inhibitorsSuccessful strategies in the discovery of small-molecule epigenetic modulators with anticancer potential.Identification of structural features of 2-alkylidene-1,3-dicarbonyl derivatives that induce inhibition and/or activation of histone acetyltransferases KAT3B/p300 and KAT2B/PCAF.Integration of Bioorthogonal Probes and Q-FRET for the Detection of Histone Acetyltransferase Activity.German-Catalan workshop on epigenetics and cancer.Comparison of transcriptomes of wild-type and isothiazolone-resistant Pseudomonas aeruginosa by using RNA-seq.Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors.Involvement of outer membrane proteins and peroxide-sensor genes in Burkholderia cepacia resistance to isothiazolone.Function-Oriented Synthesis of Marine Phidianidine Derivatives as Potential PTP1B Inhibitors with Specific Selectivity.Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 CellsPyrido- and benzisothiazolones as inhibitors of histone acetyltransferases (HATs)Rhodanine carboxylic acids as novel inhibitors of histone acetyltransferasesDesign, Synthesis, and Biological Evaluation of 2-Aminobenzanilide Derivatives as Potent and Selective HDAC Inhibitors
P2860
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P2860
Synthesis and biological testing of novel pyridoisothiazolones as histone acetyltransferase inhibitors.
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
2011年论文
@zh
2011年论文
@zh-cn
name
Synthesis and biological testi ...... acetyltransferase inhibitors.
@en
Synthesis and biological testi ...... acetyltransferase inhibitors.
@nl
type
label
Synthesis and biological testi ...... acetyltransferase inhibitors.
@en
Synthesis and biological testi ...... acetyltransferase inhibitors.
@nl
prefLabel
Synthesis and biological testi ...... acetyltransferase inhibitors.
@en
Synthesis and biological testi ...... acetyltransferase inhibitors.
@nl
P2093
P50
P1476
Synthesis and biological testi ...... acetyltransferase inhibitors.
@en
P2093
Elisabeth-Maria Bissinger
Julia M Wagner
Silviya D Furdas
Sonja Schlimme
Vassil Valkov
P304
P356
10.1016/J.BMC.2011.01.063
P407
P577
2011-02-02T00:00:00Z