Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib.
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Recent Advances in the Development and Application of Radiolabeled Kinase Inhibitors for PET ImagingCell treatment and lysis in 96-well filter-bottom plates for screening Bcr-Abl activity and inhibition in whole-cell extracts.Dosimetry of 18F-labeled tyrosine kinase inhibitor SKI-249380, a dasatinib-tracer for PET imaging.In vivo imaging of Bcr-Abl overexpressing tumors with a radiolabeled imatinib analog as an imaging surrogate for imatinib.2-18F-Fluoropropionic acid as a PET imaging agent for prostate cancer.(124)I-iodopyridopyrimidinone for PET of Abl kinase-expressing tumors in vivo.Fluorine-labeled dasatinib nanoformulations as targeted molecular imaging probes in a PDGFB-driven murine glioblastoma model.Synthesis of a [(18)F]-labeled ceritinib analogue for positron emission tomography of anaplastic lymphoma kinase, a receptor tyrosine kinase, in lung cancer.Molecular imaging for personalized cancer care.Fluorescent visualization of Src by using dasatinib-BODIPY
P2860
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P2860
Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib.
description
2007 nî lūn-bûn
@nan
2007年の論文
@ja
2007年論文
@yue
2007年論文
@zh-hant
2007年論文
@zh-hk
2007年論文
@zh-mo
2007年論文
@zh-tw
2007年论文
@wuu
2007年论文
@zh
2007年论文
@zh-cn
name
Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib.
@en
type
label
Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib.
@en
prefLabel
Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib.
@en
P2093
P356
P1476
Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib
@en
P2093
Bayard Clarkson
Blesida J Punzalan
Caryl Lambek
Darren R Veach
Elmer B Santos
Hakim Djaballah
Mohammad Namavari
Peter M Smith-Jones
Steven M Larson
Tatiana Beresten-Kochetkov
P304
P356
10.1021/JM070342G
P407
P577
2007-10-23T00:00:00Z