Naphthyl and coumarinyl biarylpiperazine derivatives as highly potent human beta-secretase inhibitors. Design, synthesis, and enzymatic BACE-1 and cell assays.
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BACE1 (β-secretase) inhibitors for the treatment of Alzheimer's disease[1,2,4]triazolo[4,3-a]phthalazines: inhibitors of diverse bromodomainsAlzheimer's disease: identification and development of β-secretase (BACE-1) binding fragments and inhibitors by dynamic ligation screening (DLS).Alzheimer's disease and mild cognitive impairmentBiological activities of guanidine compounds.Beta-secretase as a target for Alzheimer's disease drug discovery: an overview of in vitro methods for characterization of inhibitors.Synthesis, Fluorescence Properties, and Antiproliferative Potential of Several 3-Oxo-3H-benzo[f]chromene-2-carboxylic Acid Derivatives.Axonal amyloid precursor protein and its fragments undergo somatodendritic endocytosis and processing.Synthesis of novel chromene scaffolds for adenosine receptors
P2860
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P2860
Naphthyl and coumarinyl biarylpiperazine derivatives as highly potent human beta-secretase inhibitors. Design, synthesis, and enzymatic BACE-1 and cell assays.
description
2006 nî lūn-bûn
@nan
2006年の論文
@ja
2006年論文
@yue
2006年論文
@zh-hant
2006年論文
@zh-hk
2006年論文
@zh-mo
2006年論文
@zh-tw
2006年论文
@wuu
2006年论文
@zh
2006年论文
@zh-cn
name
Naphthyl and coumarinyl biaryl ...... ymatic BACE-1 and cell assays.
@en
type
label
Naphthyl and coumarinyl biaryl ...... ymatic BACE-1 and cell assays.
@en
prefLabel
Naphthyl and coumarinyl biaryl ...... ymatic BACE-1 and cell assays.
@en
P2093
P50
P356
P1476
Naphthyl and coumarinyl biaryl ...... zymatic BACE-1 and cell assays
@en
P2093
Bernard Maigret
Cédrik Garino
Gilles Quéléver
Jean-Louis Kraus
Roselyne Rosas
Takeshi Iwatsubo
Younes Laras
P304
P356
10.1021/JM0602864
P407
P577
2006-07-01T00:00:00Z