Kinetics of nonpeptide antagonist binding to the human gonadotropin-releasing hormone receptor: Implications for structure-activity relationships and insurmountable antagonism.
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Ligand binding assays at equilibrium: validation and interpretationCharacterization of 12 GnRH peptide agonists - a kinetic perspectiveDrug-target residence time--a case for G protein-coupled receptors.The Role of Target Binding Kinetics in Drug Discovery.Tactics for preclinical validation of receptor-binding radiotracers.Development of a homogeneous high-throughput live-cell G-protein-coupled receptor binding assay.Analytical method for simultaneously measuring ex vivo drug receptor occupancy and dissociation rate: application to (R)-dimethindene occupancy of central histamine H1 receptors.Triptorelin and cetrorelix induce immune responses and affect uterine development and expressions of genes and proteins of ESR1, LHR, and FSHR of mice.
P2860
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P2860
Kinetics of nonpeptide antagonist binding to the human gonadotropin-releasing hormone receptor: Implications for structure-activity relationships and insurmountable antagonism.
description
2006 nî lūn-bûn
@nan
2006年の論文
@ja
2006年論文
@yue
2006年論文
@zh-hant
2006年論文
@zh-hk
2006年論文
@zh-mo
2006年論文
@zh-tw
2006年论文
@wuu
2006年论文
@zh
2006年论文
@zh-cn
name
Kinetics of nonpeptide antagon ...... and insurmountable antagonism.
@en
type
label
Kinetics of nonpeptide antagon ...... and insurmountable antagonism.
@en
prefLabel
Kinetics of nonpeptide antagon ...... and insurmountable antagonism.
@en
P2093
P1476
Kinetics of nonpeptide antagon ...... and insurmountable antagonism.
@en
P2093
Beth A Fleck
Christopher E Heise
Paul D Crowe
R Scott Struthers
Sam R J Hoare
Susan K Sullivan
Yun-Fei Zhu
P304
P356
10.1016/J.BCP.2006.07.011
P407
P577
2006-08-22T00:00:00Z