Antitumor benzothiazoles. 3. Synthesis of 2-(4-aminophenyl)benzothiazoles and evaluation of their activities against breast cancer cell lines in vitro and in vivo.
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Models of breast cancer: is merging human and animal models the future?Indirect and direct detection of the 4-(benzothiazol-2-yl)phenylnitrenium ion from a putative metabolite of a model anti-tumor drug.Specific estrogen sulfotransferase (SULT1E1) substrates and molecular imaging probe candidates.2-[5-(Benzo[d]thia-zol-2-yl)thio-phen-2-yl]benzo[d]thia-zoleEthyl 1-[2-(morpholin-4-yl)eth-yl]-2-[4-(trifluoro-meth-yl)phen-yl]-1H-benzimid-azole-5-carboxyl-ate.Therapeutic potential of benzothiazoles: a patent review (2010 - 2014).Crystal structure of (E)-2-{[(6-meth-oxy-1,3-benzo-thia-zol-2-yl)imino]-meth-yl}phenol.Influence of 2-(4-aminophenyl)benzothiazoles on growth of human ovarian carcinoma cells in vitro and in vivo.2-(4-Aminophenyl)benzothiazoles: novel agents with selective profiles of in vitro anti-tumour activity.Mechanisms of acquired resistance to 2-(4-aminophenyl)benzothiazole (CJM 126, NSC 34445)In vitro evaluation of amino acid prodrugs of novel antitumour 2-(4-amino-3-methylphenyl)benzothiazoles.DNA damage and cell cycle arrest induced by 2-(4-amino-3-methylphenyl)-5-fluorobenzothiazole (5F 203, NSC 703786) is attenuated in aryl hydrocarbon receptor deficient MCF-7 cellsAntitumour 2-(4-aminophenyl)benzothiazoles generate DNA adducts in sensitive tumour cells in vitro and in vivoCrystal structure of the cis and trans polymorphs of bis-[μ-2-(1,3-benzo-thia-zol-2-yl)phenolato]-κ3N,O:O;κ3O:N,O-bis-[fac-tri-carbonyl-rhenium(I)].Recent advances on structural modifications of benzothiazoles and their conjugate systems as potential chemotherapeutics.Cytochrome P450 1A1-mediated anticancer drug discovery: in silico findings.Medicinal significance of benzothiazole scaffold: an insight view.Radical C-H functionalization to construct heterocyclic compounds.Antitumor activities on HL-60 human leukemia cell line, molecular docking, and quantum-chemical calculations of some sulfonamide-benzoxazoles.Synthesis and antitumor activity evaluation of new 2-(4-aminophenyl)benzothiazole derivatives bearing different heterocyclic rings.Synthesis and cytotoxic activity of 2-anilinopyridine-3-acrylamides as tubulin polymerization inhibitors.Microwave-assisted synthesis of sec/tert-butyl 2-arylbenzimidazoles and their unexpected antiproliferative activity towards ER negative breast cancer cells.3-substituted 2-phenylimidazo[2,1-b]benzothiazoles: synthesis, anticancer activity, and inhibition of tubulin polymerization.Synthesis of some N-[4-(benzothiazole-2yl) phenyl]-2-aryloxyacetamide derivatives and their anticancer activities.DNA Binding, Cleavage and Antibacterial Activity of Mononuclear Cu(II), Ni(II) and Co(II) Complexes Derived from Novel Benzothiazole Schiff Bases.N,N'-Bis(1,3-thia-zol-2-yl)methyl-ene-diamine.Characterization of the 4-(benzothiazol-2-yl)phenylnitrenium ion from a putative metabolite of a model antitumor drugChemistry of ring-substituted 4-(benzothiazol-2-yl)phenylnitrenium ions from antitumor 2-(4-aminophenyl)benzothiazoles.Synthesis, antimicrobial activity and QSAR studies of 2,5-disubstituted benzoxazoles.Novel polymer-supported coupling/dehydrating reagents for use in organic synthesis.Synthesis and Ab Initio/DFT Studies on 2-(4-methoxyphenyl)benzo[d]thiazole.Halide Control of N,N-Coordination versus N,C-Cyclometalation and Stereospecific Phenyl Ring Deuteration of Osmium(II) p-Cymene Phenylazobenzothiazole Complexes.Synthesis and antimicrobial activity of some 5-[2-(morpholin-4-yl)acetamido] and/or 5-[2-(4-substituted piperazin-1-yl)acetamido]-2-(p-substituted phenyl)benzoxazoles.Synthesis, anti-breast cancer activity, and molecular modeling of some benzothiazole and benzoxazole derivatives.Discovery of G Protein-Biased D2 Dopamine Receptor Partial Agonists.Iodine mediated oxidative cross-coupling of unprotected anilines and heteroarylation of benzothiazoles with 2-methylquinoline.Ball Milling Assisted Solvent and Catalyst Free Synthesis of Benzimidazoles and Their Derivatives.Synthesis and 11C-Radiolabelling of 2-Carboranyl Benzothiazoles.Monitoring the aggregation processes of amyloid-β using a spin-labeled, fluorescent nitroxyl radical.Excited-State Proton Transfer Can Tune the Color of Protein Fluorescent Markers.
P2860
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P2860
Antitumor benzothiazoles. 3. Synthesis of 2-(4-aminophenyl)benzothiazoles and evaluation of their activities against breast cancer cell lines in vitro and in vivo.
description
1996 nî lūn-bûn
@nan
1996年の論文
@ja
1996年論文
@yue
1996年論文
@zh-hant
1996年論文
@zh-hk
1996年論文
@zh-mo
1996年論文
@zh-tw
1996年论文
@wuu
1996年论文
@zh
1996年论文
@zh-cn
name
Antitumor benzothiazoles. 3. S ...... ll lines in vitro and in vivo.
@en
type
label
Antitumor benzothiazoles. 3. S ...... ll lines in vitro and in vivo.
@en
prefLabel
Antitumor benzothiazoles. 3. S ...... ll lines in vitro and in vivo.
@en
P2093
P356
P1476
Antitumor benzothiazoles. 3. S ...... ll lines in vitro and in vivo.
@en
P2093
Bradshaw TD
Fichtner I
Lelieveld P
Stevens MF
P304
P356
10.1021/JM9600959
P407
P577
1996-08-01T00:00:00Z