The beta-adrenergic radioligand [3H]CGP-12177, generally classified as an antagonist, is a thermogenic agonist in brown adipose tissue.
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Molecular characterization of the mouse beta 3-adrenergic receptor: relationship with the atypical receptor of adipocytesInteraction of amiodarone and triiodothyronine on the expression of beta-adrenoceptors in brown adipose tissue of ratAdrenergic stimulation of lipoprotein lipase gene expression in rat brown adipocytes differentiated in culture: mediation via beta3- and alpha1-adrenergic receptorsPharmacological approaches for the treatment of obesity.Characterization of beta 1- and beta 3-adrenoceptors in intact brown adipocytes of the rat.Atypical beta-adrenoceptors in the rat isolated common carotid arteryMetabolic response to various beta-adrenoceptor agonists in beta3-adrenoceptor knockout mice: evidence for a new beta-adrenergic receptor in brown adipose tissue.Characterization of beta-adrenoceptor mediated smooth muscle relaxation and the detection of mRNA for beta1-, beta2- and beta3-adrenoceptors in rat ileum.In situ assessment of the role of the beta 1-, beta 2- and beta 3-adrenoceptors in the control of lipolysis and nutritive blood flow in human subcutaneous adipose tissue.Mediation of most atypical effects by species homologues of the beta 3-adrenoceptor.Evidence for a functional beta 3-adrenoceptor in man.Altered sympathetic nervous system signaling in the diabetic heart: emerging targets for molecular imaging.Structural heterogeneity of membrane receptors and GTP-binding proteins and its functional consequences for signal transduction.Molecular cloning and pharmacological characterization of the bovine beta 3-adrenergic receptor.Assessment of cardiac autonomic neuronal function using PET imaging.Recent Advances and Clinical Applications of PET Cardiac Autonomic Nervous System Imaging.The biochemistry of white and brown adipocytes analysed from a selection of proteins.Beta 3- and alpha1-adrenergic Erk1/2 activation is Src- but not Gi-mediated in Brown adipocytes.Differential adrenergic regulation of the gene expression of the beta-adrenoceptor subtypes beta1, beta2 and beta3 in brown adipocytes.Evidence against beta 3-adrenoceptors or low affinity state of beta 1-adrenoceptors mediating relaxation in rat isolated aorta.Pharmacology and direct visualisation of BODIPY-TMR-CGP: a long-acting fluorescent beta2-adrenoceptor agonist.Adrenergic control of induction of type II iodothyronine 5'-deiodinase activity in cultured mouse brown adipocytes.Regulation of expression of the lipoprotein lipase gene in brown adipose tissue.β(3) Receptors: Role in Cardiometabolic Disorders.Direct demonstration of beta1- and evidence against beta2- and beta3-adrenoceptors, in smooth muscle cells of rat small mesenteric arteries.ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.Pharmacological characterization of CGP 12177 at the human beta(2)-adrenoceptor.Mechanisms of leptin secretion from white adipocytes.Radioligand binding studies of the atypical β3 -adrenergic receptor in rat brown adipose tissue using [3 H]CGP 12177
P2860
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P2860
The beta-adrenergic radioligand [3H]CGP-12177, generally classified as an antagonist, is a thermogenic agonist in brown adipose tissue.
description
1989 nî lūn-bûn
@nan
1989年の論文
@ja
1989年論文
@yue
1989年論文
@zh-hant
1989年論文
@zh-hk
1989年論文
@zh-mo
1989年論文
@zh-tw
1989年论文
@wuu
1989年论文
@zh
1989年论文
@zh-cn
name
The beta-adrenergic radioligan ...... onist in brown adipose tissue.
@en
type
label
The beta-adrenergic radioligan ...... onist in brown adipose tissue.
@en
prefLabel
The beta-adrenergic radioligan ...... onist in brown adipose tissue.
@en
P2860
P356
P1433
P1476
The beta-adrenergic radioligan ...... onist in brown adipose tissue.
@en
P2093
P2860
P304
P356
10.1042/BJ2610401
P407
P577
1989-07-01T00:00:00Z