Istaroxime stimulates SERCA2a and accelerates calcium cycling in heart failure by relieving phospholamban inhibition.
about
Phospholamban phosphorylation, mutation, and structural dynamics: a biophysical approach to understanding and treating cardiomyopathy.Sarcoendoplasmic reticulum Ca(2+) ATPase. A critical target in chlorine inhalation-induced cardiotoxicity.Novel drug targets in clinical development for heart failure.Inotropes and inodilators for acute heart failure: sarcomere active drugs in focus.New pharmacological approaches in heart failure therapy: developments and possibilities.Cardiomyocyte Ca2+ homeostasis as a therapeutic target in heart failure with reduced and preserved ejection fraction.Istaroxime, a potential anticancer drug in prostate cancer, exerts beneficial functional effects in healthy and diseased human myocardium.SERCA2a stimulation by istaroxime: a novel mechanism of action with translational implications.Conformational memory in the association of the transmembrane protein phospholamban with the sarcoplasmic reticulum calcium pump SERCA.Drug Interactions With the Ca2+-ATPase From Sarco(Endo)Plasmic Reticulum (SERCA).Correcting Calcium Dysregulation in Chronic Heart Failure Using SERCA2a Gene Therapy.Arrhythmogenic Mechanisms in Heart Failure: Linking β-Adrenergic Stimulation, Stretch, and Calcium
P2860
Q35169578-A400041E-85F9-43CA-9237-98F44C00DAA4Q35816343-6CF57ED5-663D-410F-B557-2ACE9B644623Q38202895-8DB1A726-47BC-4B05-B6AC-33628D6F1EA5Q38208442-673D3AA3-5F9E-4698-9392-8C3263728F63Q38759494-08654AC8-5DF0-4C3E-947C-AD1E2BA1DD16Q39258979-0ECDB2A8-0617-4761-8454-EF7CD70FA381Q41472411-C6D65AF2-7881-43C9-9A24-86366BC84AFAQ42014726-86761208-0A87-4B55-B144-7EEB43BBC280Q47590388-18B2FE59-6FA9-4C95-A1BA-AED90574DCBFQ52562558-6A0418AB-3FD5-4A87-8677-8592E004DF30Q52604700-B7F87805-39C7-4E67-B916-99640A2D6ED1Q58121711-806020EE-DF1F-4CD9-A7AD-26C6B694B927
P2860
Istaroxime stimulates SERCA2a and accelerates calcium cycling in heart failure by relieving phospholamban inhibition.
description
2013 nî lūn-bûn
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2013年の論文
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2013年学术文章
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2013年学术文章
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2013年学术文章
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2013年学术文章
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2013年学术文章
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name
Istaroxime stimulates SERCA2a ...... ving phospholamban inhibition.
@en
Istaroxime stimulates SERCA2a ...... ving phospholamban inhibition.
@nl
type
label
Istaroxime stimulates SERCA2a ...... ving phospholamban inhibition.
@en
Istaroxime stimulates SERCA2a ...... ving phospholamban inhibition.
@nl
prefLabel
Istaroxime stimulates SERCA2a ...... ving phospholamban inhibition.
@en
Istaroxime stimulates SERCA2a ...... ving phospholamban inhibition.
@nl
P2093
P2860
P356
P1476
Istaroxime stimulates SERCA2a ...... eving phospholamban inhibition
@en
P2093
Cristina Reina
Gianluca Bartolommei
Giuseppe Bianchi
Isabella Molinari
Mara Ferrandi
Maria Grazia Tripodi
Maria Rosa Moncelli
Paolo Barassi
Patrizia Ferrari
P2860
P304
P356
10.1111/BPH.12278
P407
P577
2013-08-01T00:00:00Z