A novel fluorescent histamine H(1) receptor antagonist demonstrates the advantage of using fluorescence correlation spectroscopy to study the binding of lipophilic ligands.

A novel fluorescent histamine H(1) receptor antagonist demonstrates the advantage of using fluorescence correlation spectroscopy to study the binding of lipophilic ligands.

Item
http://www.wikidata.org/entity/Q42058613
The evolving small-molecule fluorescent-conjugate toolbox for Class A GPCRsFluorescent approaches for understanding interactions of ligands with G protein coupled receptorsFluorescence correlation spectroscopy, combined with bimolecular fluorescence complementation, reveals the effects of β-arrestin complexes and endocytic targeting on the membrane mobility of neuropeptide Y receptorsBodilisant-a novel fluorescent, highly affine histamine h3 receptor ligandFluorescent ligands for adenosine receptors.Quantifying intracellular dynamics using fluorescence fluctuation spectroscopy.Recent applications of fluorescence correlation spectroscopy in live systems.The use of fluorescence correlation spectroscopy to characterize the molecular mobility of fluorescently labelled G protein-coupled receptors.Pharmacological Characterization of Human Histamine Receptors and Histamine Receptor Mutants in the Sf9 Cell Expression System.Use of a new proximity assay (NanoBRET) to investigate the ligand-binding characteristics of three fluorescent ligands to the human β1-adrenoceptor expressed in HEK-293 cells.High-Affinity Functional Fluorescent Ligands for Human β-Adrenoceptors.Detection of the secondary, low-affinity β1 -adrenoceptor site in living cells using the fluorescent CGP 12177 derivative BODIPY-TMR-CGP.Time-resolved fluorescence ligand binding for G protein-coupled receptors.Development of novel fluorescent histamine H1-receptor antagonists to study ligand-binding kinetics in living cells.Protein-ligand (un)binding kinetics as a new paradigm for drug discovery at the crossroad between experiments and modelling
P2860

A novel fluorescent histamine H(1) receptor antagonist demonstrates the advantage of using fluorescence correlation spectroscopy to study the binding of lipophilic ligands.

Item
http://www.wikidata.org/entity/Q42058613
description
2012 nî lūn-bûn
@nan
2012年の論文
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2012年論文
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2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
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2012年論文
@zh-tw
2012年论文
@wuu
2012年论文
@zh
2012年论文
@zh-cn
name
A novel fluorescent histamine H
@nl
A novel fluorescent histamine ...... binding of lipophilic ligands.
@en
type
label
A novel fluorescent histamine H
@nl
A novel fluorescent histamine ...... binding of lipophilic ligands.
@en
prefLabel
A novel fluorescent histamine H
@nl
A novel fluorescent histamine ...... binding of lipophilic ligands.
@en
P1433
P1476
P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P5875
P698
P932
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P1433
P1476
A novel fluorescent histamine ...... binding of lipophilic ligands.
@en
P2093
P2860
P304
P31
P356
10.1111/J.1476-5381.2011.01640.X
P407
P433
P478
P50
P577
P5875
P698
P932