about
Novel D3 selective dopaminergics incorporating enyne units as nonaromatic catechol bioisosteres: synthesis, bioactivity, and mutagenesis studiesRecent advances in the search for D3- and D4-selective drugs: probes, models and candidates.Development of Photoactivatable Allosteric Modulators for the Chemokine Receptor CXCR3.A comparison of chloroambucil- and xylene-containing polyamines leads to improved ligands for accessing the polyamine transport system.Attenuation of chemokine receptor function and surface expression as an immunomodulatory strategy employed by human cytomegalovirus is linked to vGPCR US28.Engineering a GPCR-ligand pair that simulates the activation of D(2L) by Dopamine.Cross-receptor interactions between dopamine D2L and neurotensin NTS1 receptors modulate binding affinities of dopaminergicsDiscovery of highly potent and neurotensin receptor 2 selective neurotensin mimetics.Highly potent 5-aminotetrahydropyrazolopyridines: enantioselective dopamine D3 receptor binding, functional selectivity, and analysis of receptor-ligand interactions.Dopamine D2, D3, and D4 selective phenylpiperazines as molecular probes to explore the origins of subtype specific receptor binding.The azulene framework as a novel arene bioisostere: design of potent dopamine D4 receptor ligands inducing penile erection.Identification of Two Distinct Sites for Antagonist and Biased Agonist Binding to the Human Chemokine Receptor CXCR3.Histidine 6.55 is a major determinant of ligand-biased signaling in dopamine D2L receptor.Identification of novel allosteric modulators for the G-protein coupled US28 receptor of human cytomegalovirus
P50
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P50
description
researcher
@en
wetenschapper
@nl
հետազոտող
@hy
name
Nuska Tschammer
@ast
Nuska Tschammer
@en
Nuska Tschammer
@es
Nuska Tschammer
@nl
Nuska Tschammer
@sl
type
label
Nuska Tschammer
@ast
Nuska Tschammer
@en
Nuska Tschammer
@es
Nuska Tschammer
@nl
Nuska Tschammer
@sl
prefLabel
Nuska Tschammer
@ast
Nuska Tschammer
@en
Nuska Tschammer
@es
Nuska Tschammer
@nl
Nuska Tschammer
@sl
P1053
A-7359-2008
P106
P31
P3829
P496
0000-0003-2433-3355