Novel 4'-substituted and 4',4"-disubstituted 3 alpha-(diphenylmethoxy)tropane analogs as potent and selective dopamine uptake inhibitors.
about
R-modafinil (armodafinil): a unique dopamine uptake inhibitor and potential medication for psychostimulant abuseDopamine transport inhibitors based on GBR12909 and benztropine as potential medications to treat cocaine addictionσ Receptor Effects of N-Substituted Benztropine Analogs: Implications for Antagonism of Cocaine Self-AdministrationMuscarinic preferential M(1) receptor antagonists enhance the discriminative-stimulus effects of cocaine in ratsStructure-Activity Relationships at the Monoamine Transporters for a Novel Series of Modafinil (2-[(diphenylmethyl)sulfinyl]acetamide) Analogues.Preclinical efficacy of N-substituted benztropine analogs as antagonists of methamphetamine self-administration in ratsElucidation of structural elements for selectivity across monoamine transporters: novel 2-[(diphenylmethyl)sulfinyl]acetamide (modafinil) analogues2-Substituted 3β-Aryltropane Cocaine Analogs Produce Atypical Effects without Inducing Inward-Facing Dopamine Transporter Conformations.N-substituted benztropine analogs: selective dopamine transporter ligands with a fast onset of action and minimal cocaine-like behavioral effectsProbes for the dopamine transporter: new leads toward a cocaine-abuse therapeutic--A focus on analogues of benztropine and rimcazole.Comparative structure-activity relationships of benztropine analogues at the dopamine transporter and histamine H(1) receptorsPreference for distinct functional conformations of the dopamine transporter alters the relationship between subjective effects of cocaine and stimulation of mesolimbic dopamineThe stereotypy-inducing effects of N-substituted benztropine analogs alone and in combination with cocaine do not account for their blockade of cocaine self-administration.Changes in dopamine transporter binding in nucleus accumbens following chronic self-administration cocaine: heroin combinationsRelations between stimulation of mesolimbic dopamine and place conditioning in rats produced by cocaine or drugs that are tolerant to dopamine transporter conformational change.Assessment of reinforcing effects of benztropine analogs and their effects on cocaine self-administration in rats: comparisons with monoamine uptake inhibitorsFurther delineation between typical and atypical dopamine uptake inhibitors: effects on food-maintained behavior and food consumption.Behavioral economic analysis of the effects of N-substituted benztropine analogs on cocaine self-administration in rats.Structure-Activity Relationship Studies on a Series of 3α-[Bis(4-fluorophenyl)methoxy]tropanes and 3α-[Bis(4-fluorophenyl)methylamino]tropanes As Novel Atypical Dopamine Transporter (DAT) Inhibitors for the Treatment of Cocaine Use Disorders.The Novel Modafinil Analog, JJC8-016, as a Potential Cocaine Abuse Pharmacotherapeutic.MS Binding Assays for the Three Monoamine Transporters Using the Triple Reuptake Inhibitor (1R,3S)-Indatraline as Native Marker.
P2860
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P2860
Novel 4'-substituted and 4',4"-disubstituted 3 alpha-(diphenylmethoxy)tropane analogs as potent and selective dopamine uptake inhibitors.
description
1995 nî lūn-bûn
@nan
1995年の論文
@ja
1995年論文
@yue
1995年論文
@zh-hant
1995年論文
@zh-hk
1995年論文
@zh-mo
1995年論文
@zh-tw
1995年论文
@wuu
1995年论文
@zh
1995年论文
@zh-cn
name
Novel 4'-substituted and 4',4" ...... ve dopamine uptake inhibitors.
@en
Novel 4'-substituted and 4',4" ...... ve dopamine uptake inhibitors.
@nl
type
label
Novel 4'-substituted and 4',4" ...... ve dopamine uptake inhibitors.
@en
Novel 4'-substituted and 4',4" ...... ve dopamine uptake inhibitors.
@nl
prefLabel
Novel 4'-substituted and 4',4" ...... ve dopamine uptake inhibitors.
@en
Novel 4'-substituted and 4',4" ...... ve dopamine uptake inhibitors.
@nl
P2093
P356
P1476
Novel 4'-substituted and 4',4" ...... ve dopamine uptake inhibitors.
@en
P2093
P304
P356
10.1021/JM00020A006
P407
P577
1995-09-01T00:00:00Z