Characterization of two novel sigma receptor ligands: antidystonic effects in rats suggest sigma receptor antagonism.
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Methylphenidate enhances NMDA-receptor response in medial prefrontal cortex via sigma-1 receptor: a novel mechanism for methylphenidate actionSigma receptors: potential targets for a new class of antidepressant drugIn vitro evaluation of guanidine analogs as sigma receptor ligands for potential anti-stroke therapeuticsA novel substituted piperazine, CM156, attenuates the stimulant and toxic effects of cocaine in miceThe sigma-1 antagonist BMY-14802 inhibits L-DOPA-induced abnormal involuntary movements by a WAY-100635-sensitive mechanismAn unambiguous assay for the cloned human sigma1 receptor reveals high affinity interactions with dopamine D4 receptor selective compounds and a distinct structure-affinity relationship for butyrophenonesReinforcing effects of sigma-receptor agonists in rats trained to self-administer cocaineThe dextromethorphan analog dimemorfan attenuates kainate-induced seizures via sigma1 receptor activation: comparison with the effects of dextromethorphanAntitussive activity of sigma-1 receptor agonists in the guinea-pigDifferentiation of sigma ligand-activated receptor subtypes that modulate NMDA-evoked [3H]-noradrenaline release in rat hippocampal slicesInteractions between 3,4-methylenedioxymethamphetamine and sigma1 receptorsNovel sigma (sigma) receptor agonists produce antidepressant-like effects in miceDynamic interaction between sigma-1 receptor and Kv1.2 shapes neuronal and behavioral responses to cocaineActivation of the Sigma-1 receptor by haloperidol metabolites facilitates brain-derived neurotrophic factor secretion from human astrogliaProbing the steroid binding domain-like I (SBDLI) of the sigma-1 receptor binding site using N-substituted photoaffinity labels.The Concise Guide to PHARMACOLOGY 2013/14: overview.Sigma receptor ligand, (+)-pentazocine, suppresses inflammatory responses of retinal microgliaSigma 1 receptor modulation of G-protein-coupled receptor signaling: potentiation of opioid transduction independent from receptor binding.The oligomeric states of the purified sigma-1 receptor are stabilized by ligands.Sigma-1 receptor antagonism restores injury-induced decrease of voltage-gated Ca2+ current in sensory neuronsRe-evaluation of phencyclidine low-affinity or "non-NMDA" binding sites.A role for picomolar concentrations of pregnenolone sulfate in synaptic activity-dependent Ca2+ signaling and CREB activationRelationship between cerebral sigma-1 receptor occupancy and attenuation of cocaine's motor stimulatory effects in mice by PD144418The sigma-1 receptor chaperone as an inter-organelle signaling modulatorActivation of σ-receptors induces binge-like drinking in Sardinian alcohol-preferring ratsEthanol exposure in early adolescence inhibits intrinsic neuronal plasticity via sigma-1 receptor activation in hippocampal CA1 neurons.The novel sigma-2 receptor ligand SW43 stabilizes pancreas cancer progression in combination with gemcitabine.Synthesis and pharmacological evaluation of 6-acetyl-3-(4-(4-(4-fluorophenyl)piperazin-1-yl)butyl)benzo[d]oxazol-2(3H)-one (SN79), a cocaine antagonist, in rodentsFluorescent derivatives of σ receptor ligand 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) as a tool for uptake and cellular localization studies in pancreatic tumor cells.The sigma1 receptor interacts with N-alkyl amines and endogenous sphingolipids.Intrathecal treatment with sigma1 receptor antagonists reduces formalin-induced phosphorylation of NMDA receptor subunit 1 and the second phase of formalin test in miceSynthesis and pharmacological evaluation of indole-based sigma receptor ligands.Synthesis and pharmacological characterization of a novel sigma receptor ligand with improved metabolic stability and antagonistic effects against methamphetamineEffects of UMB24 and (+/-)-SM 21, putative sigma2-preferring antagonists, on behavioral toxic and stimulant effects of cocaine in mice.The effect of the pyridyl nitrogen position in pyridylpiperazine sigma ligandsSigma-1 receptor as regulator of neuronal intracellular Ca2+: clinical and therapeutic relevance.Cocaine occupancy of sigma1 receptors and dopamine transporters in miceSigma-2 Receptors Play a Role in Cellular Metabolism: Stimulation of Glycolytic Hallmarks by CM764 in Human SK-N-SH Neuroblastoma.Synthesis and characterization of N,N-dialkyl and N-alkyl-N-aralkyl fenpropimorph-derived compounds as high affinity ligands for sigma receptors.Sigma receptors [σRs]: biology in normal and diseased states
P2860
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P2860
Characterization of two novel sigma receptor ligands: antidystonic effects in rats suggest sigma receptor antagonism.
description
1995 nî lūn-bûn
@nan
1995年の論文
@ja
1995年論文
@yue
1995年論文
@zh-hant
1995年論文
@zh-hk
1995年論文
@zh-mo
1995年論文
@zh-tw
1995年论文
@wuu
1995年论文
@zh
1995年论文
@zh-cn
name
Characterization of two novel ...... est sigma receptor antagonism.
@en
Characterization of two novel ...... est sigma receptor antagonism.
@nl
type
label
Characterization of two novel ...... est sigma receptor antagonism.
@en
Characterization of two novel ...... est sigma receptor antagonism.
@nl
prefLabel
Characterization of two novel ...... est sigma receptor antagonism.
@en
Characterization of two novel ...... est sigma receptor antagonism.
@nl
P2093
P1476
Characterization of two novel ...... est sigma receptor antagonism.
@en
P2093
P304
P356
10.1016/0014-2999(95)00208-3
P407
P577
1995-07-01T00:00:00Z