about
Base-modified Donor Analogues Reveal Novel Dynamic Features of a GlycosyltransferaseCD38 Structure-Based Inhibitor Design Using the N1-Cyclic Inosine 5'-Diphosphate Ribose TemplateCellular effects and metabolic stability of N1-cyclic inosine diphosphoribose and its derivativesSmall molecular anti-cytokine agents.New approaches to the treatment of inflammatory disorders small molecule inhibitors of p38 MAP kinase.Novel UDP-GalNAc Derivative Structures Provide Insight into the Donor Specificity of Human Blood Group Glycosyltransferase.A survey of chemical methods for sugar-nucleotide synthesis.The first C-glycosidic analogue of a novel galactosyltransferase inhibitor.Conjugation to 4-aminoquinoline improves the anti-trypanosomal activity of Deferiprone-type iron chelators.Enzymatic synthesis of nucleobase-modified UDP-sugars: scope and limitations.A novel fluorescent probe for retaining galactosyltransferases.Exploring the role of the 5-substituent for the intrinsic fluorescence of 5-aryl and 5-heteroaryl uracil nucleotides: a systematic study.Studies on the anti-inflammatory activity of phytopharmaceuticals prepared from Arnica flowers.From imidazoles to pyrimidines: new inhibitors of cytokine release.Ones, thiones, and N-oxides: an exercise in imidazole chemistry.Imidazole inhibitors of cytokine release: probing substituents in the 2 position.Identification of regioisomers in a series of N-substituted pyridin-4-yl imidazole derivatives by regiospecific synthesis, GC/MS, and 1H NMR.Novel substituted pyridinyl imidazoles as potent anticytokine agents with low activity against hepatic cytochrome P450 enzymes.Development of fluorescent aryltryptophans by Pd mediated cross-coupling of unprotected halotryptophans in water.Novel derivatives of UDP-glucose: concise synthesis and fluorescent properties.Trypanosoma brucei: chemical evidence that cathepsin L is essential for survival and a relevant drug target.Rapid synthetic route toward structurally modified derivatives of cyclic adenosine 5'-diphosphate ribose.2'-deoxy cyclic adenosine 5'-diphosphate ribose derivatives: importance of the 2'-hydroxyl motif for the antagonistic activity of 8-substituted cADPR derivatives.5-Phenyluridine trihydrate.A fast synthetic route to GDP-sugars modified at the nucleobase.Uncharged nucleoside inhibitors of β-1,4-galactosyltransferase with activity in cells.Optimised chemical synthesis of 5-substituted UDP-sugars and their evaluation as glycosyltransferase inhibitors.Base-modified NAD and AMP derivatives and their activity against bacterial DNA ligases.Rationally designed squaryldiamides – a novel class of sugar-nucleotide mimics?Two-Step Synthesis of Novel, Bioactive Derivatives of the Ubiquitous Cofactor Nicotinamide Adenine Dinucleotide (NAD)A novel fluorescent probe for NAD-consuming enzymesA facile two-step synthesis of 8-arylated guanosine mono- and triphosphates (8-aryl GXPs)Structural determinants for N1/N7 cyclization of nicotinamide hypoxanthine 5'-dinucleotide (NHD+) derivatives by ADP-ribosyl cyclase from aplysia californica: Ca2+-mobilizing activity of 8-substituted cyclic inosine 5'-diphosphoribose analogues in TInhibition of galactosyltransferases by a novel class of donor analoguesOne-step synthesis of novel glycosyltransferase inhibitorsIdentification of non-substrate-like glycosyltransferase inhibitors from library screening: pitfalls & hits
P50
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P50
description
hulumtues
@sq
onderzoeker
@nl
researcher
@en
հետազոտող
@hy
name
Gerd K. Wagner
@ast
Gerd K. Wagner
@en
Gerd K. Wagner
@es
Gerd K. Wagner
@nl
Gerd K. Wagner
@sl
type
label
Gerd K. Wagner
@ast
Gerd K. Wagner
@en
Gerd K. Wagner
@es
Gerd K. Wagner
@nl
Gerd K. Wagner
@sl
prefLabel
Gerd K. Wagner
@ast
Gerd K. Wagner
@en
Gerd K. Wagner
@es
Gerd K. Wagner
@nl
Gerd K. Wagner
@sl
P106
P1153
56321945400
P21
P31
P496
0000-0003-1086-2301