about
New approach to the practical synthesis of tri- or tetrasubstituted pyrimidine derivatives: a four-component coupling reaction from a functionalized silane, two types of aromatic nitriles, and acetals3-benzylamino-β-carboline derivatives induce apoptosis through G2/M arrest in human carcinoma cells HeLa S-3.3-(3-Phenoxybenzyl)amino-β-carboline: a novel antitumor drug targeting α-tubulin.Structure-activity relationship in the antitumor activity of 6-, 8- or 6,8-substituted 3-benzylamino-β-carboline derivatives.Determination of binding modes and binding constants for the complexes of 6H-pyrido[4,3-b]carbazole derivatives with DNA.Hf(OTf)4-catalyzed regioselective n-aminomethylation of indoles and related NH-containing heterocycles.The aminomethylation of electron-rich aromatics with an N-silyl-N,O-acetal catalyzed by a metal triflate-TMSCl system: facile synthesis of aromatic primary amines, 1-aryl-trichloroethylamines.Indium(III)-catalyzed reductive bromination and iodination of carboxylic acids to alkyl bromides and iodides: scope, mechanism, and one-pot transformation to alkyl halides and amine derivatives.An unprecedented approach to 4,5-disubstituted pyrimidine derivatives by a ZnCl(2)-catalyzed three-component coupling reaction.Palladium-catalyzed coupling reaction of terminal alkynes with aryl iodides in the presence of indium tribromide and its application to a one-pot synthesis of 2-phenylindole.Me3SiCl-promoted three-component coupling reaction of a functionalized enamine, an acetal, and an alkyne: an unprecedented approach to the synthesis of tetrasubstituted pyridines via a [3 + 2 + 1] intermolecular cyclization.InBr3-promoted divergent approach to polysubstituted indoles and quinolines from 2-ethynylanilines: switch from an intramolecular cyclization to an intermolecular dimerization by a type of terminal substituent group.Oxidative Coupling of Terminal Alkynes with Aldehydes Leading to Alkynyl Ketones by Using Indium(III) Bromide.Indium-Catalyzed Reductive Dithioacetalization of Carboxylic Acids with Dithiols: Scope, Limitations, and Application to Oxidative Desulfurization.Reductive Amination/Cyclization of Keto Acids Using a Hydrosilane for Selective Production of Lactams versus Cyclic Amines by Switching of the Indium Catalyst.Palladium-Catalyzed Reductive Coupling Reaction of Terminal Alkynes with Aryl Iodides Utilizing Hafnocene Difluoride as a Hafnium Hydride Precursor Leading to trans-Alkenes.Palladium-Catalyzed Cyclization of Alkynoic Acids To Form Vinyl Dioxanones Bearing a Quaternary Allylic Carbon.Copper-catalyzed three- five- or seven-component coupling reactions: the selective synthesis of cyanomethylamines, N,N-bis(cyanomethyl)amines and N,N'-bis(cyanomethyl)methylenediamines based on a Strecker-type synthesis.Group 4 Metallocene Difluoride/Palladium Bimetallic Catalysts for the Reductive Cross-Coupling of Alkynes with Aryl Iodides and BromidesConstruction of N-Heterocyclic Systems Containing a Fully Substituted Allylic Carbon by Palladium/Phosphine CatalysisTropene derivatives by sequential intermolecular and transannular, intramolecular palladium-catalyzed hydroamination of cycloheptatrieneNovel synthesis of 7-fluoro-8-(trifluoromethyl)- 1H-1,6-naphthyridin-4-one derivatives: intermolecular cyclization of an N-silyl-1-azaallyl anion with perfluoroalkene and subsequent intramolecular skeletal transformation of the resulting pentasubstiA single-step synthesis of enynes: Pd-catalyzed arylalkynylation of aryl iodides, internal alkynes, and alkynylsilanesDirect synthesis of polysubstituted quinoline derivatives by InBr3-promoted dimerization of 2-ethynylaniline derivativesCopper-catalyzed [5+1] annulation of 2-ethynylanilines with an N,O-acetal leading to construction of quinoline derivativesHighly selective conversion of nitrobenzenes using a simple reducing system combined with a trivalent indium salt and a hydrosilaneSynthesis of tri- or tetrasubstituted pyrimidine derivatives through the [5+1] annulation of enamidines with either N,N-dimethylformamide dialkyl acetals or orthoesters and their application in a ring transformation of pyrimidines to pyrido[2,3-d]pySingle-step thioetherification by indium-catalyzed reductive coupling of carboxylic acids with thiolsIndium-catalyzed reductive bromination of carboxylic acids leading to alkyl bromidesCopper(II)-catalyzed oxidative N-nitrosation of secondary and tertiary amines with nitromethane under an oxygen atmosphereGallium-catalyzed reductive chlorination of carboxylic acids with copper(II) chlorideIndium(III)-catalyzed knoevenagel condensation of aldehydes and activated methylenes using acetic anhydride as a promoterSynthesis and in vitro antitumor activity of novel 2-alkyl-5-methoxycarbonyl-11-methyl-6H-pyrido[4,3-b]carbazol-2-ium and 2-alkylellipticin-2-ium chloride derivativesPalladium(II)-Catalyzed Synthesis of Dibenzothiophenes from 2-Biphenylyl Disulfides by C-H FunctionalizationIndium-Catalyzed Direct Conversion of Lactones into Thiolactones Using a Disilathiane as a Sulfur SourceProduction of Quaternary α-Aminonitriles by Means of Indium-Catalyzed Three-Component Reaction of Alkynes, Amines, and Trimethylsilyl CyanidePalladium-Catalyzed Reductive Conversion of Acyl Fluorides via Ligand-Controlled DecarbonylationCatalytic C-H/C-F Coupling of Azoles and Acyl Fluorides
P50
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P50
description
Japans onderzoeker
@nl
hulumtues
@sq
investigador japonés
@es
investigador xaponés
@ast
researcher
@en
taighdeoir
@ga
հետազոտող
@hy
name
Norio Sakai
@ast
Norio Sakai
@en
Norio Sakai
@es
Norio Sakai
@nl
Norio Sakai
@sl
坂井教郎
@ja
type
label
Norio Sakai
@ast
Norio Sakai
@en
Norio Sakai
@es
Norio Sakai
@nl
Norio Sakai
@sl
坂井教郎
@ja
prefLabel
Norio Sakai
@ast
Norio Sakai
@en
Norio Sakai
@es
Norio Sakai
@nl
Norio Sakai
@sl
坂井教郎
@ja
P106
P1559
坂井教郎
@ja
P21
P27
P31
P496
0000-0003-0722-4800
P5029
read0135370
P569
2000-01-01T00:00:00Z