Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.

Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.

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http://www.wikidata.org/entity/Q44331583
Constitutive activity of the delta-opioid receptor expressed in C6 glioma cells: identification of non-peptide delta-inverse agonistsBuprenorphine/naloxone reduces the reinforcing and subjective effects of heroin in heroin-dependent volunteers.Differentiation of kappa opioid agonist-induced antinociception by naltrexone apparent pA2 analysis in rhesus monkeys.Opioid agonist efficacy predicts the magnitude of tolerance and the regulation of mu-opioid receptors and dynamin-2Most recent developments and modifications of 14-alkylamino and 14-alkoxy-4,5-epoxymorphinan derivativesHydromorphone efficacy and treatment protocol impact on tolerance and mu-opioid receptor regulation.Novel 6β-acylaminomorphinans with analgesic activity.Role of µ-opioid receptor reserve and µ-agonist efficacy as determinants of the effects of µ-agonists on intracranial self-stimulation in ratsStructural determinants of opioid activity in derivatives of 14-aminomorphinones: effect of substitution in the aromatic ring of cinnamoylaminomorphinones and codeinonesCinnamoyl derivatives of 7alpha-aminomethyl-6,14-endo-ethanotetrahydrothebaine and 7alpha-aminomethyl-6,14-endo-ethanotetrahydrooripavine and related opioid ligands.14beta-Arylpropiolylamino-17-cyclopropylmethyl-7,8-dihydronormorphinones and related opioids. Further examples of pseudoirreversible mu opioid receptor antagonists.Stratification of Cannabinoid 1 Receptor (CB1R) Agonist Efficacy: Manipulation of CB1R Density through Use of Transgenic Mice Reveals Congruence between In Vivo and In Vitro AssaysSynthesis and pharmacological evaluation of novel selective MOR agonist 6β-pyridinyl amidomorphines exhibiting long-lasting antinociception.
P2860

Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.

Item
http://www.wikidata.org/entity/Q44331583
description
1992 nî lūn-bûn
@nan
1992年の論文
@ja
1992年学术文章
@wuu
1992年学术文章
@zh
1992年学术文章
@zh-cn
1992年学术文章
@zh-hans
1992年学术文章
@zh-my
1992年学术文章
@zh-sg
1992年學術文章
@yue
1992年學術文章
@zh-hant
name
Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.
@en
Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.
@nl
type
label
Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.
@en
Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.
@nl
prefLabel
Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.
@en
Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.
@nl
P1433
P1476
P2093
P304
P31
P407
P433
P478
P577
P698
P921
P1433
P1476
Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.
@en
P2093
P304
P31
P407
P433
P478
P577
P698
P921