Novel coumarins and benzocoumarins acting as isoform-selective inhibitors against the tumor-associated carbonic anhydrase IX.
about
The anticonvulsant sulfamide JNJ-26990990 and its S,S-dioxide analog strongly inhibit carbonic anhydrases: solution and X-ray crystallographic studiesHow many carbonic anhydrase inhibition mechanisms exist?Selective inhibition of human carbonic anhydrase IX in Xenopus oocytes and MDA-MB-231 breast cancer cells.Lansoprazole and carbonic anhydrase IX inhibitors sinergize against human melanoma cells.Antitumor evaluation and molecular docking study of substituted 2-benzylidenebutane-1,3-dione, 2-hydrazonobutane-1,3-dione and trifluoromethyl-1H-pyrazole analogues.Advances in structure-based drug discovery of carbonic anhydrase inhibitors.Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase.Exploring carbonic anhydrase inhibition with multimeric coumarins displayed on a fullerene scaffold.7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring.Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors.Carbonic anhydrase inhibitors: guaiacol and catechol derivatives effectively inhibit certain human carbonic anhydrase isoenzymes (hCA I, II, IX and XII)
P2860
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P2860
Novel coumarins and benzocoumarins acting as isoform-selective inhibitors against the tumor-associated carbonic anhydrase IX.
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2013 nî lūn-bûn
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2013年学术文章
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name
Novel coumarins and benzocouma ...... ociated carbonic anhydrase IX.
@en
Novel coumarins and benzocouma ...... ociated carbonic anhydrase IX.
@nl
type
label
Novel coumarins and benzocouma ...... ociated carbonic anhydrase IX.
@en
Novel coumarins and benzocouma ...... ociated carbonic anhydrase IX.
@nl
prefLabel
Novel coumarins and benzocouma ...... ociated carbonic anhydrase IX.
@en
Novel coumarins and benzocouma ...... ociated carbonic anhydrase IX.
@nl
P2093
P2860
P1476
Novel coumarins and benzocouma ...... ociated carbonic anhydrase IX.
@en
P2093
Aditi Sharma
Claudiu T Supuran
Meena Tiwari
P2860
P304
P356
10.3109/14756366.2013.777334
P577
2013-03-14T00:00:00Z