Synthesis and antiplasmodial activity of a cysteine protease-inhibiting biotinylated aziridine-2,3-dicarboxylate.
about
Aziridine-2,3-dicarboxylate-based cysteine cathepsin inhibitors induce cell death in Leishmania major associated with accumulation of debris in autophagy-related lysosome-like vacuoles.Synthesis and biological evaluation of papain-family cathepsin L-like cysteine protease inhibitors containing a 1,4-benzodiazepine scaffold as antiprotozoal agents.Aziridine-2,3-dicarboxylates, peptidomimetic cysteine protease inhibitors with antileishmanial activity.Synthesis and molecular modeling studies of derivatives of a highly potent peptidomimetic vinyl ester as falcipain-2 inhibitors.Synthesis and evaluation of non-peptidic cysteine protease inhibitors of P. falciparum derived from etacrynic acid.Blocking effect of a biotinylated protease inhibitor on the egress of Plasmodium falciparum merozoites from infected red blood cells.Development of rhodesain inhibitors with a 3-bromoisoxazoline warhead.Structural and functional characterization of Falcipain-2, a hemoglobinase from the malarial parasite Plasmodium falciparum.
P2860
Q34309555-B4E14382-45A0-4937-92CD-993EBC400BC7Q38985765-B45D5B69-2326-4BE5-9872-57DACB60C479Q40262609-0C034C28-E8F7-4EB3-B1BB-540C83D87555Q42717133-2E206879-2BA4-422D-9BD6-8524B0F11679Q46185521-8747C7C3-A206-444A-84AB-BF48816448AFQ46520625-A45E398B-8BE1-42FE-9C66-9E13362E141AQ46636439-23A19EAE-975B-4B3D-B957-A3E27608F5A4Q48031305-331C863E-4954-4427-B47E-BFDE574F49DE
P2860
Synthesis and antiplasmodial activity of a cysteine protease-inhibiting biotinylated aziridine-2,3-dicarboxylate.
description
2004 nî lūn-bûn
@nan
2004年の論文
@ja
2004年学术文章
@wuu
2004年学术文章
@zh-cn
2004年学术文章
@zh-hans
2004年学术文章
@zh-my
2004年学术文章
@zh-sg
2004年學術文章
@yue
2004年學術文章
@zh
2004年學術文章
@zh-hant
name
Synthesis and antiplasmodial a ...... d aziridine-2,3-dicarboxylate.
@en
Synthesis and antiplasmodial a ...... d aziridine-2,3-dicarboxylate.
@nl
type
label
Synthesis and antiplasmodial a ...... d aziridine-2,3-dicarboxylate.
@en
Synthesis and antiplasmodial a ...... d aziridine-2,3-dicarboxylate.
@nl
prefLabel
Synthesis and antiplasmodial a ...... d aziridine-2,3-dicarboxylate.
@en
Synthesis and antiplasmodial a ...... d aziridine-2,3-dicarboxylate.
@nl
P2093
P2860
P356
P1433
P1476
Synthesis and antiplasmodial a ...... d aziridine-2,3-dicarboxylate.
@en
P2093
Christian L Schmidt
Christoph Gelhaus
Matthias Leippe
Radim Vicik
Rolf Hilgenfeld
P2860
P304
P356
10.1515/BC.2004.050
P577
2004-05-01T00:00:00Z