A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
about
GRL-04810 and GRL-05010, difluoride-containing nonpeptidic HIV-1 protease inhibitors (PIs) that inhibit the replication of multi-PI-resistant HIV-1 in vitro and possess favorable lipophilicity that may allow blood-brain barrier penetration.Aminofluorination of 2-alkynylanilines: a Au-catalyzed entry to fluorinated indoles.Drug metabolism in microorganisms.Recent advances in fluorination techniques and their anticipated impact on drug metabolism and toxicity.Accessing Drug Metabolites via Transition-Metal Catalyzed C-H Oxidation: The Liver as Synthetic Inspiration.Microbial biotransformation of aryl sulfanylpentafluorides.Metabolism and hydrophilicity of the polarised 'Janus face' all-cis tetrafluorocyclohexyl ring, a candidate motif for drug discovery.HIV-Associated Neurocognitive Disorder (HAND) and the Prospect of Brain-Penetrating Protease Inhibitors for Antiretroviral Treatment.Hot off the press
P2860
Q37335823-18FDE0C3-B895-4F75-B1CB-E7BB058C3351Q37619102-7C56DAD2-2D31-4BE4-8E6E-18262A7DDC5FQ38245429-DBC6382B-D203-4A51-9294-1956FA0C6056Q38366495-1F28C27B-4479-4A7A-A751-B326A27DE0EAQ38977018-5BC198EC-8593-41BA-8DAA-18BF48557EB0Q43689368-D30DF7BB-3073-4FD8-B08D-81FC38DEA3F5Q54939432-FBECCDE7-4E1F-4B33-A24D-72E4A28BFE24Q55432495-4BE0C9F7-ACAA-49C2-89A3-F4B92E96A295Q58856818-16AE5D0D-B237-4568-8C84-F3A7BBDC12CF
P2860
A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
description
2013 nî lūn-bûn
@nan
2013年の論文
@ja
2013年学术文章
@wuu
2013年学术文章
@zh
2013年学术文章
@zh-cn
2013年学术文章
@zh-hans
2013年学术文章
@zh-my
2013年学术文章
@zh-sg
2013年學術文章
@yue
2013年學術文章
@zh-hant
name
A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
@en
A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
@nl
type
label
A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
@en
A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
@nl
prefLabel
A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
@en
A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
@nl
P2093
P2860
P356
P1476
A convenient chemical-microbial method for developing fluorinated pharmaceuticals.
@en
P2093
Cormac D Murphy
Fay Dalton
Graham Sandford
Neil K O'Connor
Tara V Bright
Victoria L Elder
P2860
P304
P356
10.1039/C2OB27140K
P577
2013-02-01T00:00:00Z