A series of 2,4-disubstituted quinolines as a new class of allosteric enhancers of the adenosine A3 receptor.
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Synthesis of aryl-heteroaryl ureas (AHUs) based on 4-aminoquinoline and their evaluation against the insulin-like growth factor receptor (IGF-1R).International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and classification of adenosine receptors--an updateFunctionally biased modulation of A(3) adenosine receptor agonist efficacy and potency by imidazoquinolinamine allosteric enhancersAllosteric modulation of purine and pyrimidine receptors.Protection from myocardial ischemia/reperfusion injury by a positive allosteric modulator of the A₃ adenosine receptor.Progress towards novel adenosine receptor therapeutics gleaned from the recent patent literature.The A3 adenosine receptor as multifaceted therapeutic target: pharmacology, medicinal chemistry, and in silico approaches.Allosteric interactions at adenosine A(1) and A(3) receptors: new insights into the role of small molecules and receptor dimerization.A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy.Structure-Affinity Relationships and Structure-Kinetics Relationships of Pyrido[2,1-f]purine-2,4-dione Derivatives as Human Adenosine A3 Receptor AntagonistsSpecies differences and mechanism of action of A3 adenosine receptor allosteric modulators.A binding kinetics study of human adenosine A3 receptor agonists.Prediction of consensus binding mode geometries for related chemical series of positive allosteric modulators of adenosine and muscarinic acetylcholine receptors.
P2860
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P2860
A series of 2,4-disubstituted quinolines as a new class of allosteric enhancers of the adenosine A3 receptor.
description
2009 nî lūn-bûn
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name
A series of 2,4-disubstituted ...... of the adenosine A3 receptor.
@en
A series of 2,4-disubstituted ...... of the adenosine A3 receptor.
@nl
type
label
A series of 2,4-disubstituted ...... of the adenosine A3 receptor.
@en
A series of 2,4-disubstituted ...... of the adenosine A3 receptor.
@nl
prefLabel
A series of 2,4-disubstituted ...... of the adenosine A3 receptor.
@en
A series of 2,4-disubstituted ...... of the adenosine A3 receptor.
@nl
P2093
P50
P356
P1476
A series of 2,4-disubstituted ...... of the adenosine A3 receptor.
@en
P2093
Anikó Göblyös
Henk de Vries
Jacobus P D van Veldhoven
Johannes Brussee
Renée Bakker
Thea Mulder-Krieger
P304
P356
10.1021/JM8014052
P407
P577
2009-02-01T00:00:00Z