Selective small molecule inhibitors of the potential breast cancer marker, human arylamine N-acetyltransferase 1, and its murine homologue, mouse arylamine N-acetyltransferase 2.
about
Prospective virtual screening with Ultrafast Shape Recognition: the identification of novel inhibitors of arylamine N-acetyltransferasesArylamine N-acetyltransferases: from drug metabolism and pharmacogenetics to drug discoveryPharmGKB summary: very important pharmacogene information for N-acetyltransferase 2Piperidinols That Show Anti-Tubercular Activity as Inhibitors of Arylamine N-Acetyltransferase: An Essential Enzyme for Mycobacterial Survival Inside MacrophagesA novel color change mechanism for breast cancer biomarker detection: naphthoquinones as specific ligands of human arylamine N-acetyltransferase 1From arylamine N-acetyltransferase to folate-dependent acetyl CoA hydrolase: impact of folic acid on the activity of (HUMAN)NAT1 and its homologue (MOUSE)NAT2Identification of arylamine N-acetyltransferase inhibitors as an approach towards novel anti-tubercularsA GAA repeat expansion reporter model of Friedreich's ataxia recapitulates the genomic context and allows rapid screening of therapeutic compounds.Untargeted polar metabolomics of transformed MDA-MB-231 breast cancer cells expressing varying levels of human arylamine N-acetyltransferase 1.Crystal structure of arylamine N-acetyltransferases: insights into the mechanisms of action and substrate selectivity.Arylamine N-acetyltransferases: a structural perspective.Three-component, one-flask synthesis of rhodanines (thiazolidinones).A long-lived luminescent probe to sensitively detect arylamine N-acetyltransferase (NAT) activity of cells.Mechanisms and kinetics of human arylamine N-acetyltransferase 1 inhibition by disulfiram.Synthesis and anticancer activity of novel quinazolinone-based rhodanines.Genetic and small molecule inhibition of arylamine N-acetyltransferase 1 reduces anchorage-independent growth in human breast cancer cell line MDA-MB-231.Gold(III) chloride catalysed synthesis of 5-alkylidene-dihydrothiazoles.Metabolic activation of the cooked meat carcinogen 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine in human prostate.Comparative analysis of xenobiotic metabolising N-acetyltransferases from ten non-human primates as in vitro models of human homologues.Probing the ESIPT process in 2-amino-1,4-naphthoquinone: thermodynamics properties, solvent effect and chemometric analysisExploration of Piperidinols as Potential Antitubercular Agents
P2860
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P2860
Selective small molecule inhibitors of the potential breast cancer marker, human arylamine N-acetyltransferase 1, and its murine homologue, mouse arylamine N-acetyltransferase 2.
description
2008 nî lūn-bûn
@nan
2008年の論文
@ja
2008年学术文章
@wuu
2008年学术文章
@zh-cn
2008年学术文章
@zh-hans
2008年学术文章
@zh-my
2008年学术文章
@zh-sg
2008年學術文章
@yue
2008年學術文章
@zh
2008年學術文章
@zh-hant
name
Selective small molecule inhib ...... ylamine N-acetyltransferase 2.
@en
Selective small molecule inhib ...... ylamine N-acetyltransferase 2.
@nl
type
label
Selective small molecule inhib ...... ylamine N-acetyltransferase 2.
@en
Selective small molecule inhib ...... ylamine N-acetyltransferase 2.
@nl
prefLabel
Selective small molecule inhib ...... ylamine N-acetyltransferase 2.
@en
Selective small molecule inhib ...... ylamine N-acetyltransferase 2.
@nl
P2093
P50
P1476
Selective small molecule inhib ...... ylamine N-acetyltransferase 2.
@en
P2093
Edward D Lowe
Isaac M Westwood
James Robinson
Matthew H J Crawford
Nicola Laurieri
Stephen G Davies
P304
P356
10.1016/J.BMC.2008.11.032
P407
P577
2008-11-19T00:00:00Z