Sodium channel activators: model of binding inside the pore and a possible mechanism of action.
about
Aconitum and Delphinium sp. alkaloids as antagonist modulators of voltage-gated Na+ channels. AM1/DFT electronic structure investigations and QSAR studiesMonte Carlo-energy minimization of correolide in the Kv1.3 channel: possible role of potassium ion in ligand-receptor interactions.Action of clathrodin and analogues on voltage-gated sodium channels.Neurotoxins and their binding areas on voltage-gated sodium channels.Identification of a cluster of residues in transmembrane segment 6 of domain III of the cockroach sodium channel essential for the action of pyrethroid insecticides.Identification of new batrachotoxin-sensing residues in segment IIIS6 of the sodium channel.Batrachotoxin, pyrethroids, and BTG 502 share overlapping binding sites on insect sodium channels.Molecular biology of insect sodium channels and pyrethroid resistance.Time-dependent block and resurgent tail currents induced by mouse beta4(154-167) peptide in cardiac Na+ channels.Modular Synthesis of the Pentacyclic Core of Batrachotoxin and Select Batrachotoxin Analogue DesignsK+ channel modulators for the treatment of neurological disorders and autoimmune diseasesPiceatannol, a derivative of resveratrol, moderately slows I(Na) inactivation and exerts antiarrhythmic action in ischaemia-reperfused rat hearts.Advances in targeting voltage-gated sodium channels with small molecules.Elucidation of pyrethroid and DDT receptor sites in the voltage-gated sodium channel.The Receptor Site and Mechanism of Action of Sodium Channel Blocker Insecticides.Addition of a single methyl group to a small molecule sodium channel inhibitor introduces a new mode of gating modulation.Sodium ion unlocks understanding of channel blockadeMechanism of sodium channel block by local anesthetics, antiarrhythmics, and anticonvulsants.Structural model for dihydropyridine binding to L-type calcium channels.Inhibition of Sodium Ion Channel Function with Truncated Forms of Batrachotoxin.State-dependent inter-repeat contacts of exceptionally conserved asparagines in the inner helices of sodium and calcium channels.Structural Models of Ligand-Bound Sodium Channels.Atomic determinants of state-dependent block of sodium channels by charged local anesthetics and benzocaine.Voltage-gated Na+ channel ligands and ATP: relative molecular similarity and implications for channel function.Toxins That Affect Voltage-Gated Sodium Channels.Preliminary Results on the Evaluation of the Occurrence of Tetrodotoxin Associated to Marine Vibrio spp. in Bivalves from the Galician Rias (Northwest of Spain).Kinetic Analysis of Membrane Potential Dye Response to NaV1.7 Channel Activation Identifies Antagonists with Pharmacological Selectivity against NaV1.5.Predicting Structural Details of the Sodium Channel Pore Basing on Animal Toxin Studies
P2860
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P2860
Sodium channel activators: model of binding inside the pore and a possible mechanism of action.
description
2005 nî lūn-bûn
@nan
2005年の論文
@ja
2005年学术文章
@wuu
2005年学术文章
@zh
2005年学术文章
@zh-cn
2005年学术文章
@zh-hans
2005年学术文章
@zh-my
2005年学术文章
@zh-sg
2005年學術文章
@yue
2005年學術文章
@zh-hant
name
Sodium channel activators: mod ...... possible mechanism of action.
@en
Sodium channel activators: mod ...... possible mechanism of action.
@nl
type
label
Sodium channel activators: mod ...... possible mechanism of action.
@en
Sodium channel activators: mod ...... possible mechanism of action.
@nl
prefLabel
Sodium channel activators: mod ...... possible mechanism of action.
@en
Sodium channel activators: mod ...... possible mechanism of action.
@nl
P2860
P1433
P1476
Sodium channel activators: mod ...... possible mechanism of action.
@en
P2093
Boris S Zhorov
Denis B Tikhonov
P2860
P304
P356
10.1016/J.FEBSLET.2005.07.017
P407
P577
2005-08-01T00:00:00Z