Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
about
Macrocyclic drugs and synthetic methodologies toward macrocyclesConvergent diversity-oriented side-chain macrocyclization scan for unprotected polypeptides.Copper-catalyzed C-2 arylation or vinylation of indole derivatives with iodonium salts.Harnessing C-H Activation of Benzhydroxamates as a Macrocyclization Strategy: Synthesis of Structurally Diverse Macrocyclic Isoquinolones.Template-induced macrocycle diversity through large ring-forming alkylations of tryptophan.Mild and Regioselective Pd(OAc)2-Catalyzed C-H Arylation of Tryptophans by [ArN2]X, Promoted by Tosic Acid.New peptide architectures through C-H activation stapling between tryptophan-phenylalanine/tyrosine residuesSite-selective C(sp3)-H functionalization of di-, tri-, and tetrapeptides at the N-terminus.Palladium(II)-Catalyzed Site-Selective C(sp3 )-H Alkynylation of Oligopeptides: A Linchpin Approach for Oligopeptide-Drug Conjugation.Constrained Cyclopeptides: Biaryl Formation through Pd-Catalyzed C-H Activation in Peptides-Structural Control of the Cyclization vs. Cyclodimerization Outcome.
P2860
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P2860
Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
description
2012 nî lūn-bûn
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2012年の論文
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2012年学术文章
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2012年学术文章
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2012年学术文章
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2012年学术文章
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2012年学术文章
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2012年学术文章
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2012年學術文章
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2012年學術文章
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name
Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
@en
Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
@nl
type
label
Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
@en
Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
@nl
prefLabel
Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
@en
Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
@nl
P2093
P2860
P356
P1476
Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation.
@en
P2093
Chris Limberakis
David Price
Huijun Dong
Keith James
Spiros Liras
P2860
P304
11644-11646
P356
10.1039/C2CC36962A
P407
P577
2012-12-01T00:00:00Z