Novel vanilloid receptor-1 antagonists: 2. Structure-activity relationships of 4-oxopyrimidines leading to the selection of a clinical candidate.

Novel vanilloid receptor-1 antagonists: 2. Structure-activity relationships of 4-oxopyrimidines leading to the selection of a clinical candidate.

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http://www.wikidata.org/entity/Q46919355
Design, synthesis and biological evaluation of novel inhibitors of Trypanosoma brucei pteridine reductase 1.Mice lacking functional TRPV1 are protected from pressure overload cardiac hypertrophyTargeting Pain-evoking Transient Receptor Potential Channels for the Treatment of Pain.The thermo-TRP ion channel family: properties and therapeutic implications.Current and emerging "at-site" pain medications: a reviewCurrent perspectives on the modulation of thermo-TRP channels: new advances and therapeutic implications.Screening TRPV1 antagonists for the treatment of pain: lessons learned over a decade.Novel methodology to identify TRPV1 antagonists independent of capsaicin activation.Synthesis and cytotoxic evaluation of N-(4-methoxy-1H-benzo[d]imidazol-7-yl)-arylsulfonamide and N-aryl-(4-methoxy-1H-benzo[d]imidazol)-7-sulfonamide analogs of combretastatin A-4.Central activation of TRPV1 and TRPA1 by novel endogenous agonists contributes to mechanical allodynia and thermal hyperalgesia after burn injury.Potential Mechanisms Underlying Inflammation-Enhanced Aminoglycoside-Induced Cochleotoxicity.Heterocycle-linked phenylbenzyl amides as novel TRPV1 antagonists and their TRPV1 binding modes: constraint-induced enhancement of in vitro and in vivo activities.
P2860

Novel vanilloid receptor-1 antagonists: 2. Structure-activity relationships of 4-oxopyrimidines leading to the selection of a clinical candidate.

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http://www.wikidata.org/entity/Q46919355
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2007 nî lūn-bûn
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2007年の論文
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2007年学术文章
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2007年学术文章
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2007年学术文章
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2007年学术文章
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2007年学术文章
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2007年学术文章
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2007年學術文章
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2007年學術文章
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name
Novel vanilloid receptor-1 ant ...... ction of a clinical candidate.
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Novel vanilloid receptor-1 ant ...... ction of a clinical candidate.
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type
label
Novel vanilloid receptor-1 ant ...... ction of a clinical candidate.
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Novel vanilloid receptor-1 ant ...... ction of a clinical candidate.
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prefLabel
Novel vanilloid receptor-1 ant ...... ction of a clinical candidate.
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Novel vanilloid receptor-1 ant ...... ction of a clinical candidate.
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Novel vanilloid receptor-1 ant ...... ction of a clinical candidate.
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P2093
P304
P31
P356
P407
P433
P478
P577
P698