CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
about
Non-xanthine heterocycles: activity as antagonists of A1- and A2-adenosine receptorsPOSTER COMMUNICATIONSA 7-phenyl substituted triazolopyridazine has inverse agonist activity at the benzodiazepine receptor siteAdenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.Purine nucleosides and nucleotides as central nervous system modulators. Adenosine as the prototypic paracrine neuroactive substance.The benzodiazepine receptor.Sedative effects of PK 9084 and PK 8165, alone and in combination with chlordiazepoxideDifferential binding properties of adenosine receptor agonists and antagonists in brain.Towards functional selectivity for α6β3γ2 GABAA receptors: a series of novel pyrazoloquinolinones.Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.Modification of seizures elicited by the benzodiazepine Ro 5-3663--a comparison with picrotoxin.Photoaffinity labeling of benzodiazepine receptors in rat brain with flunitrazepam alters the affinity of benzodiazepine receptor agonist but not antagonist binding.Binding of [3H]DMCM, a convulsive benzodiazepine ligand, to rat brain membranes: preliminary studies.Development of benzodiazepine and picrotoxin (t-butylbicyclophosphorothionate) binding sites in rat cerebellar granule cells in culture.The biological basis of benzodiazepine actions.Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.Aminophylline and CGS 8216 reverse the protective action of diazepam against electroconvulsions in mice.Benzodiazepine receptor antagonists reverse the effect of diazepam on plasma corticosterone in stressed rats.Poster Communications
P2860
Q24599034-0172FC61-C82D-4B15-ABAA-1EDF528C9C71Q29031985-D393FB11-513A-4EF5-B66E-05450196968CQ35887671-EFA7DB83-B4B9-4E49-8ED1-78A33230C7F3Q36332205-88E7554E-A238-49EB-9293-391D65F23EFDQ37610889-94E7C5DA-F231-4E73-8736-CCAB697C4A74Q39505550-2B916C2B-3BB3-43B2-BA81-742F82151186Q41830694-E66A881D-ACEE-4974-8EAD-94DC75E28CB7Q42246465-73F77868-EA0F-42B2-88A5-CE3D1CF01D53Q47974409-CD5503D7-CFEA-41F5-9D8E-7CED0DA51B8FQ48433873-0AEE8E96-4FEA-424C-948A-B69916615148Q48660653-2C55D085-99C2-46C9-B519-3254C5E782F6Q48722047-414129CA-6DA1-4814-A28F-3A5DFD2602F9Q48771378-E5E4BE13-5CDA-4478-B6EF-5CE1BE143120Q49116678-33C524BB-05D7-43E7-854C-AF86572C2675Q51245870-174118C3-84FE-4CE2-8C71-1200B825E7BBQ51765905-DF91B44F-419B-443E-90AB-906E03B43674Q51820343-B0EEC041-0CC2-4E17-BFC2-636C2408825BQ51848572-5F1939A7-E8B8-4F23-9715-79F7DDD5D313Q58830772-9F015699-54D8-48A9-88E6-354A393636FD
P2860
CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
description
1982 nî lūn-bûn
@nan
1982年の論文
@ja
1982年学术文章
@wuu
1982年学术文章
@zh
1982年学术文章
@zh-cn
1982年学术文章
@zh-hans
1982年学术文章
@zh-my
1982年学术文章
@zh-sg
1982年學術文章
@yue
1982年學術文章
@zh-hant
name
CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
@en
CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
@nl
type
label
CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
@en
CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
@nl
prefLabel
CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
@en
CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
@nl
P2093
P1433
P1476
CGS 8216: receptor binding characteristics of a potent benzodiazepine antagonist.
@en
P2093
Brundish DE
Czernik AJ
Kalinsky HJ
Psychoyos S
Rinehart RK
P304
P356
10.1016/0024-3205(82)90573-2
P407
P577
1982-01-01T00:00:00Z