about
The metal face of protein tyrosine phosphatase 1BSmall molecule inhibitors of West Nile virus.Parallel synthesis of "click" chalcones as antitubulin agents.Solution-phase parallel synthesis of aryloxyimino amides via a novel multicomponent reaction among aromatic (Z)-chlorooximes, isocyanides, and electron-deficient phenols.The tubulin colchicine domain: a molecular modeling perspective.Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus.Haptic-driven applications to molecular modeling: state-of-the-art and perspectives.Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: Synthesis and biological evaluation.Solution-phase parallel synthesis and biological evaluation of combretatriazoles.Crystal structure of human nicotinic acid phosphoribosyltransferase.Descriptive structure-separation relationship studies in chiral ligand-exchange chromatography.Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs.Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity.Zinc ions modulate protein tyrosine phosphatase 1B activity.ZINClick: a database of 16 million novel, patentable, and readily synthesizable 1,4-disubstituted triazoles.Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors.Broad tuning of the human bitter taste receptor hTAS2R46 to various sesquiterpene lactones, clerodane and labdane diterpenoids, strychnine, and denatonium.Rational Discovery of (+) (S) Abscisic Acid as a Potential Antifungal Agent: a Repurposing Approach.De novo computer-aided design of novel antiviral agentsDesign, Synthesis, and Biological Evaluation of Combretabenzodiazepines: A Novel Class of Anti-Tubulin AgentsAre 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups?A Practical Synthesis of 5-Aroyl-1-aryltetrazoles Using an Ugi-Like 4-Component Reaction Followed by a Biomimetic TransaminationEstrogenic Analogues Synthesized by Click ChemistryDiscovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to in Vivo Pharmacodynamic ActivitySynthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 InhibitorsPhotocatalytic Isocyanide-Based Multicomponent Domino Cascade toward the Stereoselective Formation of IminofuransZINClick v.18: Expanding Chemical Space of 1,2,3-TriazolesBio-Inspired Dual-Selective BCL-2/c-MYC G-Quadruplex Binders: Design, Synthesis, and Anticancer Activity of Drug-like Imidazo[2,1-i]purine DerivativesEssential Medicinal Chemistry of Essential Medicines
P50
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P50
description
onderzoeker
@nl
researcher
@en
հետազոտող
@hy
name
Alberto Massarotti
@ast
Alberto Massarotti
@en
Alberto Massarotti
@es
Alberto Massarotti
@nl
Alberto Massarotti
@sl
type
label
Alberto Massarotti
@ast
Alberto Massarotti
@en
Alberto Massarotti
@es
Alberto Massarotti
@nl
Alberto Massarotti
@sl
prefLabel
Alberto Massarotti
@ast
Alberto Massarotti
@en
Alberto Massarotti
@es
Alberto Massarotti
@nl
Alberto Massarotti
@sl
P1053
O-8293-2015
P106
P1153
24577732200
P21
P31
P3829
P496
0000-0001-9306-8845