Synthesis, pharmacological evaluation and conformational investigation of endomorphin-2 hybrid analogues

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Structural and biological exploration of phe(3)-phe(4)-modified endomorphin-2 peptidomimetics.Endomorphin-1 analogs containing α-methyl-β-amino acids exhibit potent analgesic activity after peripheral administration.

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Q39779368-470F224D-B490-4732-9DFE-4B22AD5E0BBE Q52092987-BB241ECB-C3A1-4D1F-984D-B9C59F7BD490

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Synthesis, pharmacological evaluation and conformational investigation of endomorphin-2 hybrid analogues

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im November 2012 veröffentlichter wissenschaftlicher Artikel

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wetenschappelijk artikel

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наукова стаття, опублікована в листопаді 2012

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Synthesis, pharmacological eva ...... endomorphin-2 hybrid analogues

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Synthesis, pharmacological eva ...... endomorphin-2 hybrid analogues

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Synthesis, pharmacological eva ...... endomorphin-2 hybrid analogues

@en

Synthesis, pharmacological eva ...... endomorphin-2 hybrid analogues

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Synthesis, pharmacological eva ...... endomorphin-2 hybrid analogues

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Synthesis, pharmacological eva ...... endomorphin-2 hybrid analogues

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Synthesis, pharmacological eva ...... endomorphin-2 hybrid analogues

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Anna Borsodi

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Engin Bojnik

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Francesco Airaghi

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Gianfranco Balboni

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Giordano Lesma

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Teresa Recca

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Functional Selectivity and Classical Concepts of Quantitative Pharmacology

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Environmental mimic of receptor interaction: conformational analysis of CCK-15 in solution.

Further studies on lead compounds containing the opioid pharmacophore Dmt-Tic.

Synthesis and evaluation of new endomorphin-2 analogues containing (Z)-alpha,beta-didehydrophenylalanine (Delta(Z)Phe) residues.

Endomorphin-1 and endomorphin-2: pharmacology of the selective endogenous mu-opioid receptor agonists.

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s11030-012-9399-5

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19-31

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scholarly article

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10.1007/S11030-012-9399-5

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P478

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Severo Salvadori

Alessandra Silvani

Alessandro Sacchetti

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2012-11-04T00:00:00Z

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23124951

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Farmakologi

Synthesis, pharmacological evaluation and conformational investigation of endomorphin-2 hybrid analogues

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Synthesis, pharmacological evaluation and conformational investigation of endomorphin-2 hybrid analogues

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P1476

P2093

P2860

P2888

P304

P31

P356

P433

P478

P50

P577

P698

P921

P356

P1433

P1476

P2093

P2860

P2888

P304

P31

P356

P433

P478

P50

P577

P698

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