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Nicotinic acetylcholine receptor ligands, a patent review (2006-2011)Prenylated indole alkaloids from Flustra foliacea with subtype specific binding on NAChRsSynthesis and nicotinic binding studies on enantiopure diazine analogues of the novel (2-chloro-5-pyridyl)-9-azabicyclo[4.2.1]non-2-ene UB-165.Semisynthetic analogues of toxiferine I and their pharmacological properties at α7 nAChRs, muscle-type nAChRs, and the allosteric binding site of muscarinic M2 receptors.Smoking upregulates alpha4beta2* nicotinic acetylcholine receptors in the human brain.The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor ligands. Part 2: carboxamide derivatives with different spacer motifs.The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor (nAChR) ligands. Part 1: the influence of different hydrogen bond acceptor systems on alkyl and (hetero)aryl substituents.Nicotine decreases food intake through activation of POMC neurons.The twin drug approach for novel nicotinic acetylcholine receptor ligands.Carbazole Scaffold in Medicinal Chemistry and Natural Products: A Review from 2010-2015.Bispidine as a Privileged Scaffold.Feasibility of [18F]-2-Fluoro-A85380-PET imaging of human vascular nicotinic acetylcholine receptors in vivoCytisine-based nicotinic partial agonists as novel antidepressant compounds.A hydrazide linker strategy for heterobivalent compounds as ortho- and allosteric ligands of acetylcholine-binding proteins.Syntheses and evaluation of pyridazine and pyrimidine containing bioisosteres of (+/-)-pyrido[3.4-b]homotropane and pyrido-[3.4-b]tropane as novel nAChR ligands.3D QSAR analyses-guided rational design of novel ligands for the (alpha4)2(beta2)3 nicotinic acetylcholine receptor.Synthesis and evaluation of phenylcarbamate derivatives as ligands for nicotinic acetylcholine receptors.In vitro characterization of 6-[18F]fluoro-A-85380, a high-affinity ligand for alpha4beta2* nicotinic acetylcholine receptors.Halogenated and isosteric cytisine derivatives with increased affinity and functional activity at nicotinic acetylcholine receptors.Effects of Abeta1-42 fibrils and of the tetrapeptide Pr-IIGL on the phosphorylation state of the tau-protein and on the alpha7 nicotinic acetylcholine receptor in vitro.6H,13H-Pyrazino[1,2-a;4,5-a']diindole analogs: probing the pharmacophore for allosteric ligands of muscarinic M2 receptors.Heliotropiumides A and B, new phenolamides with N-carbamoyl putrescine moiety from Heliotropium foertherianum collected in Hawaii and their biological activities.In vitro evaluation of nicotinic acetylcholine receptors with 2-[18F]F-A85380 in Parkinson's disease.Synthetic approaches and bio-distribution studies of [11C]methyl-phenidate.Feasibility of 2-deoxy-2-[18F]fluoro-D-glucose- A85380-PET for imaging of human cardiac nicotinic acetylcholine receptors in vivo.[Nuclides and tracers--mechanisms and application. Radiodiagnosis for peripheral organ diseases].Development of a 5-Hydroxytryptamine2A Receptor Binding Assay for High Throughput Screening Using 96-Well Microfilter Plates
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P50
name
Daniela Gündisch
@en
Daniela Gündisch
@nl
type
label
Daniela Gündisch
@en
Daniela Gündisch
@nl
prefLabel
Daniela Gündisch
@en
Daniela Gündisch
@nl