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Q39807616-C53A5D35-D08B-43BC-84E4-2F6F358F5FE3
Q39807616-C53A5D35-D08B-43BC-84E4-2F6F358F5FE3
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Statement
http://www.wikidata.org/entity/statement/Q39807616-C53A5D35-D08B-43BC-84E4-2F6F358F5FE3
Nilotinib concentration in cell lines and primary CD34(+) chronic myeloid leukemia cells is not mediated by active uptake or efflux by major drug transporters.
P2860
Q39807616-C53A5D35-D08B-43BC-84E4-2F6F358F5FE3
BestRank
Statement
http://www.wikidata.org/entity/statement/Q39807616-C53A5D35-D08B-43BC-84E4-2F6F358F5FE3
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wasDerivedFrom
8617ce4eb14732f742085e2a0372cd2bf09a1480
P2860
OCT-1-mediated influx is a key determinant of the intracellular uptake of imatinib but not nilotinib (AMN107): reduced OCT-1 activity is the cause of low in vitro sensitivity to imatinib