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Q55242399-9742EE4D-EB12-4301-85BC-BA2CD5497E4F
Q55242399-9742EE4D-EB12-4301-85BC-BA2CD5497E4F
BestRank
Statement
http://www.wikidata.org/entity/statement/Q55242399-9742EE4D-EB12-4301-85BC-BA2CD5497E4F
Specific stereochemistry of OP-1074 disrupts estrogen receptor alpha helix 12 and confers pure antiestrogenic activity.
P2860
Q55242399-9742EE4D-EB12-4301-85BC-BA2CD5497E4F
BestRank
Statement
http://www.wikidata.org/entity/statement/Q55242399-9742EE4D-EB12-4301-85BC-BA2CD5497E4F
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Statement
wasDerivedFrom
fc21bbe4df270753ef5c4a4791a3b20f7350eedb
P2860
The turnover of estrogen receptor α by the selective estrogen receptor degrader (SERD) fulvestrant is a saturable process that is not required for antagonist efficacy