Pharmacological characterization of membrane-expressed human trace amine-associated receptor 1 (TAAR1) by a bioluminescence resonance energy transfer cAMP biosensor - Test2 - elhamkhani - TriplyDB

Pharmacological characterization of membrane-expressed human trace amine-associated receptor 1 (TAAR1) by a bioluminescence resonance energy transfer cAMP biosensor

Pharmacological characterization of membrane-expressed human trace amine-associated receptor 1 (TAAR1) by a bioluminescence resonance energy transfer cAMP biosensor

http://www.wikidata.org/entity/Q24627304

about

The dopamine metabolite 3-methoxytyramine is a neuromodulator Trace amine-associated receptors as emerging therapeutic targets The emerging role of trace amine-associated receptor 1 in the functional regulation of monoamine transporters and dopaminergic activity Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class International Union of Pharmacology. LXXII. Recommendations for trace amine receptor nomenclature Trace Amines and the Trace Amine-Associated Receptor 1: Pharmacology, Neurochemistry, and Clinical Implications Genetically-encoded tools for cAMP probing and modulation in living systems Methamphetamine and HIV-1-induced neurotoxicity: role of trace amine associated receptor 1 cAMP signaling in astrocytes Determinants involved in subtype-specific functions of rat trace amine-associated receptors 1 and 4 Cyclic AMP control measured in two compartments in HEK293 cells: phosphodiesterase K(M) is more important than phosphodiesterase localization The role of GRK6 in animal models of Parkinson's disease and L-DOPA treatment Human and mouse trace amine-associated receptor 1 have distinct pharmacology towards endogenous monoamines and imidazoline receptor ligands.Bariatric endocrinology: principles of medical practice.Pharmacological characterization of a small-molecule agonist for the chemokine receptor CXCR3 Decoy receptor CXCR7 modulates adrenomedullin-mediated cardiac and lymphatic vascular development.Functional interaction between trace amine-associated receptor 1 and dopamine D2 receptor Biased signaling at chemokine receptors Avenues for the development of therapeutics that target trace amine associated receptor 1 (TAAR1).BRET Biosensor Analysis of Receptor Tyrosine Kinase Functionality.Antagonism of dopamine D2 receptor/beta-arrestin 2 interaction is a common property of clinically effective antipsychotics.Triphenylmethane dye activation of beta-arrestin BRET biosensors to study GPCR biology, pharmacology, and signal transduction.Biophysical techniques for detection of cAMP and cGMP in living cells.Integrated approaches to understanding antipsychotic drug action at GPCRs.Modulation of Glucagon-like Peptide-1 (GLP-1) Potency by Endocannabinoid-like Lipids Represents a Novel Mode of Regulating GLP-1 Receptor Signaling.Tyramine and β-phenylethylamine, from fermented food products, as agonists for the human trace amine-associated receptor 1 (hTAAR1) in the stomach.Role of SAP97 protein in the regulation of corticotropin-releasing factor receptor 1 endocytosis and extracellular signal-regulated kinase 1/2 signaling TAAR1-dependent effects of apomorphine in mice.Adenylyl cyclase activating polypeptide reduces phosphorylation and toxicity of the polyglutamine-expanded androgen receptor in spinobulbar muscular atrophy.MAGI Proteins Regulate the Trafficking and Signaling of Corticotropin-Releasing Factor Receptor 1 via a Compensatory Mechanism.The Case for TAAR1 as a Modulator of Central Nervous System Function.Characterization of Dopaminergic System in the Striatum of Young Adult Park2-/- Knockout Rats.Increased trace amine-associated receptor 1 (TAAR1) expression is associated with a positive survival rate in patients with breast cancer.Further insights into the pharmacology of the human trace amine-associated receptors: discovery of novel ligands for TAAR1 by a virtual screening approach.Insights into the structure and pharmacology of the human trace amine-associated receptor 1 (hTAAR1): homology modelling and docking studies.The Trace Amine-Associated Receptor 1 Agonist 3-Iodothyronamine Induces Biased Signaling at the Serotonin 1b Receptor.Intracellular cAMP Sensor EPAC: Physiology, Pathophysiology, and Therapeutics Development.A cAMP Biosensor-Based High-Throughput Screening Assay for Identification of Gs-Coupled GPCR Ligands and Phosphodiesterase Inhibitors.TAAR1 induces a disturbed GSK3β phosphorylation in recurrent miscarriages through the ODC.Biochemical and Functional Characterization of the Trace Amine-Associated Receptor 1 (TAAR1) Agonist RO5263397.

P2860

Q21091097-CE146E46-4D8D-47C0-8FD3-6D871CE09244 Q22242286-35A52604-277C-4DDA-A85E-013A9A7A2B5B Q22242368-6168D004-A848-406A-A4BA-1107589D8349 Q22252340-E9983104-0480-411D-A7A8-28893A67F8A2 Q24634650-B948997C-F9F0-4099-BDBB-EB3C907A12AB Q26752602-1F52F6BD-920C-491D-AA4C-35EE6EE6017B Q26781567-B3EE2BAB-BB6C-4B86-9F12-FB4E1DE0AFF0 Q28242470-4DC3F062-AE7D-4716-8083-736B3803E351 Q28704020-83FA2486-EAC0-498B-A1BF-9F9A91978EDC Q28740548-017A4304-ECFE-4E62-9CB2-5A3D79F137C0 Q30506209-7E73703F-1EC7-4451-8054-976C0456C06C Q33499502-8903C176-2AEE-412A-9C79-070B32AB2882 Q33677790-EE04BE33-F4A1-4CAF-A604-5F111EFF7C85 Q34007358-DF9FDADD-591F-41F1-B183-217AB181F866 Q34199625-E8071DE1-C5C7-418D-B0A8-EA60CEF0F112 Q35188101-FA653E65-D3EC-4EF6-B2F4-66C6E4510E9A Q35351711-BD3C764C-D485-405C-98E2-59B15C1BA4EC Q36746446-EAF1216F-5A01-4080-B7E8-2524A7C093C4 Q36750306-729CFB99-F4DA-4B1D-98F3-FEFEC25B1EB7 Q36870038-51AC82C6-D078-4422-8F54-9C475395A3EB Q37096786-0B40171A-FB73-4DCA-A1BF-FA540FA26A34 Q38041105-7B51A70F-7AF9-407A-9E1E-53F46AD87797 Q38098831-10D32752-6364-4838-8702-1044FBFACA8F Q38200335-7A125C9E-35D2-45BA-9749-036EB5A42B5D Q38883453-225DB451-F222-4F1D-9BC5-A26840EB77A6 Q39022680-BB4937E7-6A23-488E-8719-36FEBF1974FE Q41018207-5217B9EE-4637-433E-93B1-489B13AAF0BE Q45743520-34B4BA6B-0031-4A03-811C-35D049D91843 Q46025171-F97EA801-013F-4D8A-99E7-19357247F4F5 Q46335711-7DF2817A-AD6C-4FBB-AF2E-B0874A57DDCC Q47640093-2AABB74D-9372-4C8E-94ED-17221FDA2C9B Q48171776-3E5AFEEF-1CE0-492A-BCC7-0D2F753B954B Q48275344-AAF6B92B-D573-4B2A-8A0F-78FE009A3108 Q48281018-9301D868-B111-4DDD-A8A2-967E3C914FA8 Q48413428-234596E2-6350-4513-BF18-F3DF6B7BE868 Q51733160-ED64F31E-7A13-4D97-ADC1-C599FE23046B Q52656382-D26F65C9-E04A-4E75-84EA-9D1E0AA71043 Q53551796-92A0AF9F-3B17-4BCE-AD2D-EAF7A18ACCAB Q54124939-2303D06C-94BF-42E1-9453-5720D76790AC Q55446730-40D779F5-E65A-4CEE-A7A7-10D7D28789C0

P2860

Pharmacological characterization of membrane-expressed human trace amine-associated receptor 1 (TAAR1) by a bioluminescence resonance energy transfer cAMP biosensor

http://www.wikidata.org/entity/Q24627304

description

2008 nî lūn-bûn

@nan

2008 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած

@hyw

2008 թվականի սեպտեմբերին հրատարակված գիտական հոդված

@hy

2008年の論文

@ja

2008年論文

@yue

2008年論文

@zh-hant

2008年論文

@zh-hk

2008年論文

@zh-mo

2008年論文

@zh-tw

2008年论文

@wuu

name

Pharmacological characterizati ...... energy transfer cAMP biosensor

@ast

Pharmacological characterizati ...... energy transfer cAMP biosensor

@en

Pharmacological characterizati ...... energy transfer cAMP biosensor

@nl

type

label

Pharmacological characterizati ...... energy transfer cAMP biosensor

@ast

Pharmacological characterizati ...... energy transfer cAMP biosensor

@en

Pharmacological characterizati ...... energy transfer cAMP biosensor

@nl

prefLabel

Pharmacological characterizati ...... energy transfer cAMP biosensor

@ast

Pharmacological characterizati ...... energy transfer cAMP biosensor

@en

Pharmacological characterizati ...... energy transfer cAMP biosensor

@nl

P1433

Q24627304-088A0244-DA4E-429A-90D3-572FE269D420

P1476

Q24627304-E1B32FAD-B48A-4638-A89C-D3A39F55250D

P2093

Q24627304-18892878-4C47-4D91-AC9A-5B8C03712914

Q24627304-36F5F0B8-6AE5-4BED-8C28-823CD1249CAD

Q24627304-3B1C4C51-2CFD-45F8-9993-468BA12DBFB1

Q24627304-642A4964-5D57-4B51-82DF-FA795A318085

Q24627304-6CB79DEB-5A03-4FDB-AA03-655F806660CC

Q24627304-7D47D17A-8A10-4098-A951-518F9014ADF8

Q24627304-CBE4BC1A-3E09-477D-ACDE-CD87BD3380EA

P2860

Q24627304-055E5A51-C48B-49C8-9600-8655A4DB99FF

Q24627304-08A9284C-58EF-4280-8166-8BC7A924AD42

Q24627304-11494506-294C-4F9A-A709-BA946C236757

Q24627304-1913334A-A881-4D0F-AAF2-A340E8EA531A

Q24627304-1ACBA892-96BA-45CE-8515-716B2E9C22E4

Q24627304-21D61308-BF8A-4864-974A-67B31F838455

Q24627304-2A65E16B-FC4F-4B59-B9F1-0FF6DCF6A320

Q24627304-3943058E-49EC-49F5-A32C-66A897D11FA8

Q24627304-415DDF37-22AD-42D2-860D-7727E347E1DF

Q24627304-42FC6418-68AE-4BDB-9911-96366C6C2B90

P304

Q24627304-5D8FE065-8237-4B16-A545-15EBAA46448F

P31

Q24627304-4AB03FB0-0B26-4727-B807-8075995BB1A9

P3181

Q24627304-113B7831-B378-4060-97DF-3C5B3E2E630A

P356

Q24627304-C6AD0E17-0E9F-4835-80D7-A2AAF767BA26

P407

Q24627304-73EF58BA-A948-43C6-9EAE-EF4C6BF64EBE

P433

Q24627304-3DE48DDE-2A12-48B1-909C-388FB3C877D7

P478

Q24627304-7B20D106-3A04-40F1-B116-C6FC9687CB72

P50

Q24627304-5A966C05-A682-41B0-B370-990AE247182C

Q24627304-61826828-70E0-4BF8-B5FE-135CA7D70732

Q24627304-6C0D81E6-CC75-4D1A-98A8-1C78CABAF492

P577

Q24627304-3F0F4E46-DB06-4E80-9A13-A345320086D1

P5875

Q24627304-BF8BE0D5-7DB4-48D2-8365-35CED7CF62D4

P698

Q24627304-6115E756-3766-47F8-B17D-05B2232BC3A6

P921

Q24627304-2B011F42-B9EC-4EEE-A065-7EBCF50FABE9

Q24627304-7CD29656-3772-4C00-889A-D40633A5C02F

Q24627304-D918CA35-C147-4C54-ACB3-6BC688168093

P932

Q24627304-DC9A9C34-1A6E-4835-9565-0844AFCD3F40

P3181

P356

P1433

Molecular Pharmacology

P1476

Pharmacological characterizati ...... energy transfer cAMP biosensor

@en

P2093

Ali Salahpour

http://www.w3.org/2001/XMLSchema#string

Jonathan D Violin

http://www.w3.org/2001/XMLSchema#string

Larry S Barak

http://www.w3.org/2001/XMLSchema#string

Marc G Caron

http://www.w3.org/2001/XMLSchema#string

Robert J Lefkowitz

http://www.w3.org/2001/XMLSchema#string

Tatyana D Sotnikova

http://www.w3.org/2001/XMLSchema#string

Xiaodong Zhang

http://www.w3.org/2001/XMLSchema#string

P2860

A renaissance in trace amines inspired by a novel GPCR family

L-DOPA: From a biologically inactive amino acid to a successful therapeutic agent

Amphetamine, 3,4-methylenedioxymethamphetamine, lysergic acid diethylamide, and metabolites of the catecholamine neurotransmitters are agonists of a rat trace amine receptor

RTP family members induce functional expression of mammalian odorant receptors

Trace amines: identification of a family of mammalian G protein-coupled receptors

Trace amine-associated receptor 1-Family archetype or iconoclast?

Cell physiology of cAMP sensor Epac.

A beta-arrestin/green fluorescent protein biosensor for detecting G protein-coupled receptor activation

3-Iodothyronamine is an endogenous and rapid-acting derivative of thyroid hormone

Mechanisms of amphetamine action revealed in mice lacking the dopamine transporter

P304

585-594

http://www.w3.org/2001/XMLSchema#string

P31

scholarly article

P3181

2471220

http://www.w3.org/2001/XMLSchema#string

P356

10.1124/MOL.108.048884

http://www.w3.org/2001/XMLSchema#string

P407

P433

3

http://www.w3.org/2001/XMLSchema#string

P478

74

http://www.w3.org/2001/XMLSchema#string

P50

Raul Gainetdinov

P577

2008-06-04T00:00:00Z

http://www.w3.org/2001/XMLSchema#dateTime

P5875

51401184

http://www.w3.org/2001/XMLSchema#string

P698

18524885

http://www.w3.org/2001/XMLSchema#string

P921

bioluminescence

biosensing technique

P932

3766527

http://www.w3.org/2001/XMLSchema#string