Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
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Small-molecule Binding to the DNA Minor Groove Is Mediated by a Conserved Water ClusterStructure-in vitro activity relationships of pentamidine analogues and dication-substituted bis-benzimidazoles as new antifungal agentsIn vitro antifungal activities of a series of dication-substituted carbazoles, furans, and benzimidazolesCombined treatment of heterocyclic analogues and benznidazole upon Trypanosoma cruzi in vivoPharmacology of DB844, an orally active aza analogue of pafuramidine, in a monkey model of second stage human African trypanosomiasisHighly active anti-Pneumocystis carinii compounds in a library of novel piperazine-linked bisbenzamidines and related compounds.Arylimidamide DB766, a potential chemotherapeutic candidate for Chagas' disease treatment(E)-1,1'-Bis[(E)-but-2-en-yl]-3,3'-(propane-1,3-di-yl)bis-(1H-benzimidazol-3-ium) dibromide monohydrate.In vitro selection and in vivo efficacy of piperazine- and alkanediamide-linked bisbenzamidines against Pneumocystis pneumonia in mice.CYP4F enzymes are the major enzymes in human liver microsomes that catalyze the O-demethylation of the antiparasitic prodrug DB289 [2,5-bis(4-amidinophenyl)furan-bis-O-methylamidoxime].Human African trypanosomiasis: pharmacological re-engagement with a neglected disease.Antiparasitic compounds that target DNA.Efficacy of the novel diamidine compound 2,5-Bis(4-amidinophenyl)- furan-bis-O-Methlylamidoxime (Pafuramidine, DB289) against Trypanosoma brucei rhodesiense infection in vervet monkeys after oral administration.Neglected disease - african sleeping sickness: recent synthetic and modeling advances.Water-mediated binding of agents that target the DNA minor groove.Quantitative analysis of amphiphilic N-alkyloxypyridinecarboximidamide by liquid chromatography-tandem mass spectrometry.
P2860
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P2860
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
description
1998 nî lūn-bûn
@nan
1998 թուականի Մարտին հրատարակուած գիտական յօդուած
@hyw
1998 թվականի մարտին հրատարակված գիտական հոդված
@hy
1998年の論文
@ja
1998年論文
@yue
1998年論文
@zh-hant
1998年論文
@zh-hk
1998年論文
@zh-mo
1998年論文
@zh-tw
1998年论文
@wuu
name
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs
@nl
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
@ast
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
@en
type
label
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs
@nl
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
@ast
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
@en
prefLabel
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs
@nl
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
@ast
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
@en
P2093
P2860
P1476
Anti-Pneumocystis activities of aromatic diamidoxime prodrugs.
@en
P2093
B C Bender
D A Patrick
J E Kerrigan
J P Stanko
K Ramachandran
R R Tidwell
P2860
P304
P407
P577
1998-03-01T00:00:00Z