The comparative pharmacology and up-regulation of rat neuronal nicotinic receptor subtype binding sites stably expressed in transfected mammalian cells
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Phantasmidine: an epibatidine congener from the ecuadorian poison frog Epipedobates anthonyiMammalian nicotinic acetylcholine receptors: from structure to functionTranslational research in nicotine dependenceLow dose nicotine and antagonism of β2 subunit containing nicotinic acetylcholine receptors have similar effects on affective behavior in miceQuantitative analysis of the heteromeric neuronal nicotinic receptors in the rat hippocampusNicotinic receptor subunit alpha5 modifies assembly, up-regulation, and response to pro-inflammatory cytokines[(3)H]Epibatidine photolabels non-equivalent amino acids in the agonist binding site of Torpedo and alpha4beta2 nicotinic acetylcholine receptorsCognitive deficits in schizophrenia: focus on neuronal nicotinic acetylcholine receptors and smoking.Developmental effects of acute, chronic, and withdrawal from chronic nicotine on fear conditioning.The alpha 3 subunit gene of the nicotinic acetylcholine receptor is a candidate gene for ethanol stimulationNocturnal frontal lobe epilepsy with paroxysmal arousals due to CHRNA2 loss of functionCholine promotes nicotinic receptor alpha4 + beta2 up-regulationPolyethylene glycol-based homologated ligands for nicotinic acetylcholine receptorsCharacterizing low affinity epibatidine binding to α4β2 nicotinic acetylcholine receptors with ligand depletion and nonspecific bindingAlexa Fluor 546-ArIB[V11L;V16A] is a potent ligand for selectively labeling alpha 7 nicotinic acetylcholine receptorsAT-1001: a high affinity and selective α3β4 nicotinic acetylcholine receptor antagonist blocks nicotine self-administration in rats.Drug discrimination in methamphetamine-trained rats: effects of cholinergic nicotinic compounds.Oxidative folding and preparation of α-conotoxins for use in high-throughput structure-activity relationship studies.Increased nicotinic acetylcholine receptor protein underlies chronic nicotine-induced up-regulation of nicotinic agonist binding sites in mouse brainDiscovery of a potent and selective α3β4 nicotinic acetylcholine receptor antagonist from an α-conotoxin synthetic combinatorial library.Effects of chronic nicotine on heteromeric neuronal nicotinic receptors in rat primary cultured neurons.Pharmacological stress is required for the anti-alcohol effect of the α3β4* nAChR partial agonist AT-1001Endogenously expressed muscarinic receptors in HEK293 cells augment up-regulation of stably expressed α4β2 nicotinic receptors.Upregulation of Nicotinic Acetylcholine Receptor alph4+beta2 through a Ligand-Independent PI3Kbeta Mechanism That Is Enhanced by TNFalpha and the Jak2/p38Mapk Pathways.Menthol Enhances the Desensitization of Human α3β4 Nicotinic Acetylcholine Receptors.AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors.Regulation of the distribution and function of [(125)I]epibatidine binding sites by chronic nicotine in mouse embryonic neuronal culturesChronic sazetidine-A at behaviorally active doses does not increase nicotinic cholinergic receptors in rodent brain.Neuronal nicotinic acetylcholine receptor expression and function on nonneuronal cells.Competition, Selectivity and Efficacy of Analogs of A-84543 for Nicotinic Acetylcholine Receptors with Repositioning of Pyridine Nitrogen.Synthesis and pharmacological evaluation of novel 9- and 10-substituted cytisine derivatives. Nicotinic ligands of enhanced subtype selectivity.Muscle and neuronal nicotinic acetylcholine receptors. Structure, function and pathogenicity.Gene targeting demonstrates that alpha4 nicotinic acetylcholine receptor subunits contribute to expression of diverse [3H]epibatidine binding sites and components of biphasic 86Rb+ efflux with high and low sensitivity to stimulation by acetylcholineIdentifying the lipid-protein interface of the alpha4beta2 neuronal nicotinic acetylcholine receptor: hydrophobic photolabeling studies with 3-(trifluoromethyl)-3-(m-[125I]iodophenyl)diazirine.Divergent functional effects of sazetidine-a and varenicline during nicotine withdrawal.Genetic background influences the effects of withdrawal from chronic nicotine on learning and high-affinity nicotinic acetylcholine receptor binding in the dorsal and ventral hippocampusChemistry and pharmacological studies of 3-alkoxy-2,5-disubstituted-pyridinyl compounds as novel selective α4β2 nicotinic acetylcholine receptor ligands that reduce alcohol intake in ratsSynthesis and biological evaluation of novel carbon-11 labeled pyridyl ethers: candidate ligands for in vivo imaging of alpha4beta2 nicotinic acetylcholine receptors (alpha4beta2-nAChRs) in the brain with positron emission tomography[¹²⁵I]AT-1012, a new high affinity radioligand for the α3β4 nicotinic acetylcholine receptors.Evidence from mouse and man for a role of neuregulin 3 in nicotine dependence.
P2860
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P2860
The comparative pharmacology and up-regulation of rat neuronal nicotinic receptor subtype binding sites stably expressed in transfected mammalian cells
description
2004 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2004 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
artículu científicu espublizáu en 2004
@ast
im Juli 2004 veröffentlichter wissenschaftlicher Artikel
@de
scientific journal article
@en
vedecký článok (publikovaný 2004/07/01)
@sk
vědecký článek publikovaný v roce 2004
@cs
wetenschappelijk artikel (gepubliceerd op 2004/07/01)
@nl
наукова стаття, опублікована в липні 2004
@uk
مقالة علمية (نشرت في يوليو 2004)
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name
The comparative pharmacology a ...... in transfected mammalian cells
@ast
The comparative pharmacology a ...... in transfected mammalian cells
@en
The comparative pharmacology a ...... in transfected mammalian cells
@nl
type
label
The comparative pharmacology a ...... in transfected mammalian cells
@ast
The comparative pharmacology a ...... in transfected mammalian cells
@en
The comparative pharmacology a ...... in transfected mammalian cells
@nl
prefLabel
The comparative pharmacology a ...... in transfected mammalian cells
@ast
The comparative pharmacology a ...... in transfected mammalian cells
@en
The comparative pharmacology a ...... in transfected mammalian cells
@nl
P356
P1476
The comparative pharmacology a ...... in transfected mammalian cells
@en
P2093
Kenneth J. Kellar
Yingxian Xiao
P304
P356
10.1124/JPET.104.066787
P407
P577
2004-07-01T00:00:00Z