Design, synthesis and interaction at the vesicular monoamine transporter-2 of lobeline analogs: potential pharmacotherapies for the treatment of psychostimulant abuse.
about
Novel N-1,2-dihydroxypropyl analogs of lobelane inhibit vesicular monoamine transporter-2 function and methamphetamine-evoked dopamine release.Modeling in vitro inhibition of butyrylcholinesterase using molecular docking, multi-linear regression and artificial neural network approachesN-terminus regulation of VMAT2 mediates methamphetamine-stimulated efflux.Synthesis of Lobeline, Lobelane and their Analogues. A Review.Exploring the effect of N-substitution in nor-lobelane on the interaction with VMAT2: discovery of a potential clinical candidate for treatment of methamphetamine abuse.Lobelane analogues containing 4-hydroxy and 4-(2-fluoroethoxy) aromatic substituents: Potent and selective inhibitors of [(3)H]dopamine uptake at the vesicular monoamine transporter-2.1,4-Diphenalkylpiperidines: A new scaffold for the design of potent inhibitors of the vesicular monoamine transporter-2.
P2860
Q34202539-AEB2B142-94E1-4CC7-937D-CFB1748432ACQ37574117-116A7D3A-A920-4DF5-A8AE-E6CC83687181Q37589110-4087FDE0-1DFB-4B97-9393-FE1D1F5A80AEQ38267226-4B681CBF-FA50-4035-9696-2D8E0EBACE13Q42098885-F1837E14-C95B-48BB-A7CF-63DA809DE97AQ42373565-497A6190-3543-4EA6-85E4-36F7CB72E1B1Q42418144-DA2FBC22-40EA-4C33-B3F0-6E11344DE735
P2860
Design, synthesis and interaction at the vesicular monoamine transporter-2 of lobeline analogs: potential pharmacotherapies for the treatment of psychostimulant abuse.
description
2011 nî lūn-bûn
@nan
2011 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Design, synthesis and interact ...... ment of psychostimulant abuse.
@ast
Design, synthesis and interact ...... ment of psychostimulant abuse.
@en
type
label
Design, synthesis and interact ...... ment of psychostimulant abuse.
@ast
Design, synthesis and interact ...... ment of psychostimulant abuse.
@en
prefLabel
Design, synthesis and interact ...... ment of psychostimulant abuse.
@ast
Design, synthesis and interact ...... ment of psychostimulant abuse.
@en
P2093
P2860
P1476
Design, synthesis and interact ...... ment of psychostimulant abuse.
@en
P2093
Ashish P Vartak
David B Horton
Fang Zheng
Guangrong Zheng
John P Culver
Linda P Dwoskin
Peter A Crooks
P2860
P304
P356
10.2174/156802611795371332
P577
2011-01-01T00:00:00Z