An efficient high-throughput screening method for MYST family acetyltransferases, a new class of epigenetic drug targets.

An efficient high-throughput screening method for MYST family acetyltransferases, a new class of epigenetic drug targets.

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http://www.wikidata.org/entity/Q34075283
Progress in epigenetic histone modification analysis by mass spectrometry for clinical investigationsHistone-modifying enzymes, histone modifications and histone chaperones in nucleosome assembly: Lessons learned from Rtt109 histone acetyltransferasesA cell-free fluorometric high-throughput screen for inhibitors of Rtt109-catalyzed histone acetylationComputational Analysis and Predictive Cheminformatics Modeling of Small Molecule Inhibitors of Epigenetic ModifiersA powerful yeast-based screening assay for the identification of inhibitors of indoleamine 2,3-dioxygenase.The essential roles of chemistry in high-throughput screening triagePAINS in the assay: chemical mechanisms of assay interference and promiscuous enzymatic inhibition observed during a sulfhydryl-scavenging HTS.MOZ regulates B-cell progenitors and, consequently, Moz haploinsufficiency dramatically retards MYC-induced lymphoma development.Crosstalk between epigenetic readers regulates the MOZ/MORF HAT complexes.Chromatin modifiers and the promise of epigenetic therapy in acute leukemiaChemical Biology for Investigating Epigenetic Functions of Lysine Acetyltransferases (KATs).Expression of the MOZ-TIF2 oncoprotein in mice represses senescenceAssay interference and off-target liabilities of reported histone acetyltransferase inhibitors.Uncovering a novel pathway for p16 silencing: Therapeutic implications for lung cancer.Seven Year Itch: Pan-Assay Interference Compounds (PAINS) in 2017-Utility and Limitations.New KAT6 inhibitors induce senescence and arrest cancer growth
P2860

An efficient high-throughput screening method for MYST family acetyltransferases, a new class of epigenetic drug targets.

Item
http://www.wikidata.org/entity/Q34075283
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2011 nî lūn-bûn
@nan
2011 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
An efficient high-throughput s ...... ss of epigenetic drug targets.
@ast
An efficient high-throughput s ...... ss of epigenetic drug targets.
@en
An efficient high-throughput s ...... ss of epigenetic drug targets.
@nl
type
label
An efficient high-throughput s ...... ss of epigenetic drug targets.
@ast
An efficient high-throughput s ...... ss of epigenetic drug targets.
@en
An efficient high-throughput s ...... ss of epigenetic drug targets.
@nl
prefLabel
An efficient high-throughput s ...... ss of epigenetic drug targets.
@ast
An efficient high-throughput s ...... ss of epigenetic drug targets.
@en
An efficient high-throughput s ...... ss of epigenetic drug targets.
@nl
P1433
P1476
P2093
P2860
P304
P31
P356
P433
P478
P50
P577
P5875
P698
P921
P356
P1433
P1476
An efficient high-throughput s ...... ss of epigenetic drug targets.
@en
P2093
P2860
P304
P31
P356
P433
P478
P50
P577
P5875
P698
P921