Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
about
Neurosteroids and GABA(A) Receptor Interactions: A Focus on StressThe anti-convulsant stiripentol acts directly on the GABA(A) receptor as a positive allosteric modulatorAntagonism of neurosteroid modulation of native gamma-aminobutyric acid receptors by (3alpha,5alpha)-17-phenylandrost-16-en-3-olGABAA receptor-acting neurosteroids: a role in the development and regulation of the stress responseNeurosteroids: endogenous regulators of the GABA(A) receptorAllopregnanolone in the bed nucleus of the stria terminalis modulates contextual fear in rats.Neuroactive steroid stereospecificity of ethanol-like discriminative stimulus effects in monkeys.Cyclodextrins sequester neuroactive steroids and differentiate mechanisms that rate limit steroid actionsMidazolam inhibits hippocampal long-term potentiation and learning through dual central and peripheral benzodiazepine receptor activation and neurosteroidogenesis.Treatment with and withdrawal from finasteride alter ethanol intake patterns in male C57BL/6J mice: potential role of endogenous neurosteroids?The effect of age on the discriminative stimulus effects of ethanol and its GABA(A) receptor mediation in cynomolgus monkeys.Flavan-3-ol esters: new agents for exploring modulatory sites on GABA(A) receptors.Neurosteroids and GABA-A Receptor Function.A 17beta-derivative of allopregnanolone is a neurosteroid antagonist at a cerebellar subpopulation of GABA A receptors with nanomolar affinity.Mechanisms of neurosteroid interactions with GABA(A) receptors.Mechanisms of potentiation of the mammalian GABAA receptor by the marine cembranoid eupalmerin acetateNeurosteroids, stress and depression: potential therapeutic opportunities.Comparison of Steroid Modulation of Spontaneous Inhibitory Postsynaptic Currents in Cultured Hippocampal Neurons and Steady-State Single-Channel Currents from Heterologously Expressed α1β2γ2L GABA(A) Receptors.Mutations of the GABA-A receptor alpha1 subunit M1 domain reveal unexpected complexity for modulation by neuroactive steroids.The influence of neuroactive steroid lipophilicity on GABAA receptor modulation: evidence for a low-affinity interaction.Neurosteroid interactions with synaptic and extrasynaptic GABA(A) receptors: regulation of subunit plasticity, phasic and tonic inhibition, and neuronal network excitability.Photodynamic effects of steroid-conjugated fluorophores on GABAA receptors.Acute and chronic effects of ethanol on learning-related synaptic plasticity.Microtubule ionic conduction and its implications for higher cognitive functions.A mutant residue in the third transmembrane region of the GABA(A) alpha1 subunit causes increased agonistic neurosteroid responses.Novel Molecule Exhibiting Selective Affinity for GABAA Receptor Subtypes.A spontaneous tonic chloride conductance in solitary glutamatergic hippocampal neurons.Intrathecal neurosteroids and a neurosteroid antagonist: effects on inflammation-evoked thermal hyperalgesia and tactile allodynia.Modulating GABA modulators.Neurosteroids involved in regulating inhibition in the inferior colliculus.
P2860
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P2860
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
description
2004 nî lūn-bûn
@nan
2004 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2004 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2004年の論文
@ja
2004年論文
@yue
2004年論文
@zh-hant
2004年論文
@zh-hk
2004年論文
@zh-mo
2004年論文
@zh-tw
2004年论文
@wuu
name
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA
@nl
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
@ast
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
@en
type
label
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA
@nl
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
@ast
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
@en
prefLabel
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA
@nl
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
@ast
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
@en
P2093
P356
P1476
Selective antagonism of 5alpha-reduced neurosteroid effects at GABA(A) receptors.
@en
P2093
Alex S Evers
Amanda Shute
Brad D Manion
Charles F Zorumski
Douglas F Covey
Mingde Wang
Steven Mennerick
P304
P356
10.1124/MOL.65.5.1191
P577
2004-05-01T00:00:00Z