Cell-based systems to assess nuclear receptor activation and their use in drug development.
about
Marine invertebrate xenobiotic-activated nuclear receptors: their application as sensor elements in high-throughput bioassays for marine bioactive compoundsPregnane X receptor and drug-induced liver injury.A novel approach applying a chemical biology strategy in phenotypic screening reveals pathway-selective regulators of histone 3 K27 tri-methylation.Size does matter! Label-free detection of small molecule-protein interaction.Advantages of cell-based high-volume screening assays to assess nuclear receptor activation during drug discovery.Mechanisms of xenobiotic receptor activation: Direct vs. indirect.CYP3A4-dependent cellular response does not relate to CYP3A4-catalysed metabolites of C-1748 and C-1305 acridine antitumor agents in HepG2 cells.
P2860
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P2860
Cell-based systems to assess nuclear receptor activation and their use in drug development.
description
2013 nî lūn-bûn
@nan
2013 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
name
Cell-based systems to assess n ...... their use in drug development.
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Cell-based systems to assess n ...... their use in drug development.
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Cell-based systems to assess n ...... their use in drug development.
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Cell-based systems to assess n ...... their use in drug development.
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Cell-based systems to assess n ...... their use in drug development.
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Cell-based systems to assess n ...... their use in drug development.
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Cell-based systems to assess n ...... their use in drug development.
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Cell-based systems to assess n ...... their use in drug development.
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Cell-based systems to assess n ...... their use in drug development.
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P2860
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Cell-based systems to assess n ...... their use in drug development.
@en
P2093
Jerome M Lasker
Judy L Raucy
P2860
P304
P356
10.3109/03602532.2012.737333
P407
P577
2013-02-01T00:00:00Z