Ginkgolide B and bilobalide block the pore of the 5-HT₃receptor at a location that overlaps the picrotoxin binding site

Ginkgolide B and bilobalide block the pore of the 5-HT₃receptor at a location that overlaps the picrotoxin binding site

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http://www.wikidata.org/entity/Q34762077
The Concise Guide to PHARMACOLOGY 2013/14: ligand-gated ion channels.Neuroprotective effects of bilobalide on cerebral ischemia and reperfusion injury are associated with inhibition of pro-inflammatory mediator production and down-regulation of JNK1/2 and p38 MAPK activation.Binding sites for bilobalide, diltiazem, ginkgolide, and picrotoxinin at the 5-HT3 receptor.Noncompetitive Inhibition of 5-HT3 Receptors by Citral, Linalool, and Eucalyptol Revealed by Nonlinear Mixed-Effects Modeling.Advantages of an antagonist: bicuculline and other GABA antagonists.Discriminating between 5-HT₃A and 5-HT₃AB receptorsCysteine modification reveals which subunits form the ligand binding site in human heteromeric 5-HT3AB receptors.A golden approach to ion channel inhibitionFunctional Brain Activity Changes after 4 Weeks Supplementation with a Multi-Vitamin/Mineral Combination: A Randomized, Double-Blind, Placebo-Controlled Trial Exploring Functional Magnetic Resonance Imaging and Steady-State Visual Evoked Potentials dTricyclic antidepressant amitriptyline inhibits 5-hydroxytryptamine 3 receptor currents in NCB-20 cells
P2860

Ginkgolide B and bilobalide block the pore of the 5-HT₃receptor at a location that overlaps the picrotoxin binding site

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http://www.wikidata.org/entity/Q34762077
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2010 nî lūn-bûn
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2010 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
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2010 թվականի նոյեմբերին հրատարակված գիտական հոդված
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2010年の論文
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2010年学术文章
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2010年学术文章
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2010年学术文章
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Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@ast
Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@en
Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@nl
type
label
Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@ast
Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@en
Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@nl
prefLabel
Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@ast
Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@en
Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@nl
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P5875
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Ginkgolide B and bilobalide bl ...... ps the picrotoxin binding site
@en
P2093
P2860
P304
P31
P356
10.1016/J.NEUROPHARM.2010.11.003
P433
P478
P577
P5875
P698
P932