A new-generation 5-nitroimidazole can induce highly metronidazole-resistant Giardia lamblia in vitro.
about
Drug Development Against the Major Diarrhea-Causing Parasites of the Small Intestine, Cryptosporidium and GiardiaDrug Resistance in the Microaerophilic Parasite Giardia lambliaStructural and functional perturbation of Giardia lamblia triosephosphate isomerase by modification of a non-catalytic, non-conserved regionA rapid, high-throughput viability assay for Blastocystis spp. reveals metronidazole resistance and extensive subtype-dependent variations in drug susceptibilities.High-throughput Giardia lamblia viability assay using bioluminescent ATP content measurementsA reprofiled drug, auranofin, is effective against metronidazole-resistant Giardia lambliaPyruvate:ferredoxin oxidoreductase and thioredoxin reductase are involved in 5-nitroimidazole activation while flavin metabolism is linked to 5-nitroimidazole resistance in Giardia lambliaImpaired parasite attachment as fitness cost of metronidazole resistance in Giardia lamblia.Antigiardial activity of novel triazolyl-quinolone-based chalcone derivatives: when oxygen makes the difference.Click Chemistry-Facilitated Structural Diversification of Nitrothiazoles, Nitrofurans, and Nitropyrroles Enhances Antimicrobial Activity against Giardia lamblia.O(2)-dependent efficacy of novel piperidine- and piperazine-based chalcones against the human parasite Giardia intestinalis.Understanding drug resistance in human intestinal protozoa.The past, present and future of fluorescent protein tags in anaerobic protozoan parasites.In vitro antigiardial activity of the cysteine protease inhibitor E-64.In vitro activity of the F-6 fraction of oregano against Giardia intestinalis.An Efficient One-Pot Catalyzed Synthesis of 2,4-Disubstituted 5-Nitroimidazoles Displaying Antiparasitic and Antibacterial Activities.Reconstruction of Sugar Metabolic Pathways of Giardia lamblia.Metabolism of nitro drugs metronidazole and nitazoxanide in Giardia lamblia: characterization of a novel nitroreductase (GlNR2).TDAE strategy in the benzoxazolone series: synthesis and reactivity of a new benzoxazolinonic anion.A review on metronidazole: an old warhorse in antimicrobial chemotherapy.Differential protein expression and post-translational modifications in metronidazole-resistant Giardia duodenalis.Nitroreductase (GlNR1) increases susceptibility of Giardia lamblia and Escherichia coli to nitro drugs.
P2860
Q26774724-2B9BCDCA-4AC7-4BED-B492-C47FB571EB24Q26800010-049BC9BC-9113-4FFD-9579-385C7269BFE3Q27679239-8AEBF9F0-D460-4E64-B2E1-7349BCF326DBQ34528996-A8500AE5-46D2-4F86-B9ED-D01775924470Q34529169-9651F4FE-788F-4211-8B6E-1ABDDF6AD80EQ34583468-25CC0829-7AB8-4913-821E-DAD9A5D520ECQ35096900-1F026F22-C327-4D01-90CE-158170A0A012Q35270323-BDE81B75-22CC-40EB-83C7-F6D5E0C92832Q35315705-9755DEB7-06A1-4B92-883C-6CB3A963F782Q36342610-17A4F923-24E3-44BC-A755-92551B225AA3Q37544469-9CA3DBED-C025-414C-B38F-42C8E15ACA1DQ38381784-54228223-74C3-4FA9-BD98-58C94F4FF957Q38665237-4EF62C10-642C-46F1-872D-5327B2007453Q39247809-75AC69B7-8C2B-4DA5-8FA7-450DC06CEE05Q39656013-1C30B70D-B48E-4531-9EF7-0057837B2AF0Q40108442-FCE349F1-DD52-43C5-ADCC-52B88F864F04Q41643525-00089FAC-36A3-4395-8BD7-B650D0EF5A0FQ45219788-89DD52C6-6AF4-44EC-86D6-6870AA3950C4Q46832754-16F325E8-9573-4BE2-AC8A-7B693A0C97DAQ49790580-6253DCBB-F4CF-4D55-B809-CD3AEE30D1A3Q52567256-D5DD977C-3DC2-445B-8F21-62D2D298738EQ54365687-D7E21D98-B1E9-4C1D-9142-F21C391CF5DA
P2860
A new-generation 5-nitroimidazole can induce highly metronidazole-resistant Giardia lamblia in vitro.
description
2010 nî lūn-bûn
@nan
2010 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
A new-generation 5-nitroimidaz ...... tant Giardia lamblia in vitro.
@ast
A new-generation 5-nitroimidaz ...... tant Giardia lamblia in vitro.
@en
type
label
A new-generation 5-nitroimidaz ...... tant Giardia lamblia in vitro.
@ast
A new-generation 5-nitroimidaz ...... tant Giardia lamblia in vitro.
@en
prefLabel
A new-generation 5-nitroimidaz ...... tant Giardia lamblia in vitro.
@ast
A new-generation 5-nitroimidaz ...... tant Giardia lamblia in vitro.
@en
P2093
P2860
P1476
A new-generation 5-nitroimidaz ...... tant Giardia lamblia in vitro.
@en
P2093
Anita G Burgess
Frances D Gillin
Jacqueline A Upcroft
Kenia G Krauer
Lars Eckmann
Linda A Dunn
Maxime D Crozet
Patrice Vanelle
Peter Upcroft
P2860
P356
10.1016/J.IJANTIMICAG.2010.03.004
P577
2010-04-24T00:00:00Z