about
Polymyxins and quinazolines are LSD1/KDM1A inhibitors with unusual structural featuresAssessing histone demethylase inhibitors in cells: lessons learned.Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells.Chemical probes targeting epigenetic proteins: Applications beyond oncology.Small molecules targeting histone demethylase genes (KDMs) inhibit growth of temozolomide-resistant glioblastoma cellsChoose and Use Your Chemical Probe Wisely to Explore Cancer Biology.Highly selective inhibition of histone demethylases by de novo macrocyclic peptides.Advances toward LSD1 inhibitors for cancer therapy.Novel potent inhibitors of the histone demethylase KDM1A (LSD1), orally active in a murine promyelocitic leukemia model.Inhibitors of Protein Methyltransferases and Demethylases.4-Biphenylalanine- and 3-Phenyltyrosine-Derived Hydroxamic Acids as Inhibitors of the JumonjiC-Domain-Containing Histone Demethylase KDM4A.Epigenetic gene regulation by histone demethylases: emerging role in oncogenesis and inflammation.The molecular underpinnings of prostate cancer: impacts on management and pathology practice.Epigenetic Treatment of Persistent Viral Infections.Design of KDM4 Inhibitors with Antiproliferative Effects in Cancer Models.Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7.Two-State Reactivity of Histone Demethylases Containing Jumonji-C Active Sites: Different Mechanisms for Different Methylation Degrees.Structure-Based Design of a New Scaffold for Cell-Penetrating Peptidic Inhibitors of the Histone Demethylase PHF8.Compounds and methods for inhibiting histone demethylases: a patent evaluation of US20160102096A1.Inhibitors of both the N-methyl lysyl- and arginyl-demethylase activities of the JmjC oxygenases.The Emerging Role of Histone Demethylases in Renal Cell Carcinoma.Targeting Cancer with PCPA-Drug Conjugates: LSD1 Inhibition-Triggered Release of 4-Hydroxytamoxifen.JMJD5 is a human arginyl C-3 hydroxylase.Small molecule KDM4s inhibitors as anti-cancer agents.Mechanistic and structural studies of KDM-catalysed demethylation of histone 1 isotype 4 at lysine 26Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7
P2860
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P2860
description
2015 nî lūn-bûn
@nan
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
2015年论文
@zh
2015年论文
@zh-cn
name
Recent Progress in Histone Demethylase Inhibitors.
@ast
Recent Progress in Histone Demethylase Inhibitors.
@en
type
label
Recent Progress in Histone Demethylase Inhibitors.
@ast
Recent Progress in Histone Demethylase Inhibitors.
@en
prefLabel
Recent Progress in Histone Demethylase Inhibitors.
@ast
Recent Progress in Histone Demethylase Inhibitors.
@en
P50
P1476
Recent Progress in Histone Demethylase Inhibitors.
@en
P2093
Katherine S England
P304
P356
10.1021/ACS.JMEDCHEM.5B01758
P407
P577
2015-12-28T00:00:00Z