about
Molecular and functional properties of P2X receptors--recent progress and persisting challengesCrystal structure of the ATP-gated P2X(4) ion channel in the closed stateInsights into the channel gating of P2X receptors from structures, dynamics and small moleculesSize matters in activation/inhibition of ligand-gated ion channelsSolution structure of the rat P2X4 receptor head domain involved in inhibitory metal binding.Alpha-hemolysin from Escherichia coli uses endogenous amplification through P2X receptor activation to induce hemolysis.A P2X receptor from the tardigrade species Hypsibius dujardini with fast kinetics and sensitivity to zinc and copper.Sphingosine-1-phosphate elicits receptor-dependent calcium signaling in retinal amacrine cellsPannexin-1 hemichannel-mediated ATP release together with P2X1 and P2X4 receptors regulate T-cell activation at the immune synapse.Gintonin, a ginseng-derived lysophosphatidic acid receptor ligand, potentiates ATP-gated P2X₁ receptor channel currentsCloning and characterization of a P2X receptor expressed in the central nervous system of Lymnaea stagnalisActivation and regulation of purinergic P2X receptor channelsThe P2X1 ion channel in platelet function.New structure enlivens interest in P2X receptors.Structural interpretation of P2X receptor mutagenesis studies on drug actionKey sites for P2X receptor function and multimerization: overview of mutagenesis studies on a structural basis.Suppression of cell membrane permeability by suramin: involvement of its inhibitory actions on connexin 43 hemichannels.Amitriptyline does not block the action of ATP at human P2X4 receptor.Molecular basis of selective antagonism of the P2X1 receptor for ATP by NF449 and suramin: contribution of basic amino acids in the cysteine-rich loop.Use of chimeras, point mutants, and molecular modeling to map the antagonist-binding site of 4,4',4″,4‴-(carbonylbis-(imino-5,1,3-benzenetriylbis(carbonylimino)))tetrakisbenzene-1,3-disulfonic acid (NF449) at P2X1 receptors for ATP.P2X receptor chimeras highlight roles of the amino terminus to partial agonist efficacy, the carboxyl terminus to recovery from desensitization, and independent regulation of channel transitions
P2860
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P2860
description
2008 nî lūn-bûn
@nan
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
2008年论文
@zh
2008年论文
@zh-cn
name
Ectodomain lysines and suramin block of P2X1 receptors.
@en
Ectodomain lysines and suramin block of P2X1 receptors.
@nl
type
label
Ectodomain lysines and suramin block of P2X1 receptors.
@en
Ectodomain lysines and suramin block of P2X1 receptors.
@nl
prefLabel
Ectodomain lysines and suramin block of P2X1 receptors.
@en
Ectodomain lysines and suramin block of P2X1 receptors.
@nl
P2093
P2860
P356
P1476
Ectodomain lysines and suramin block of P2X1 receptors.
@en
P2093
Helen E Broomhead
Joan A Sim
R Alan North
P2860
P304
29841-29846
P356
10.1074/JBC.M802523200
P407
P577
2008-09-02T00:00:00Z